Progress in the Development of Non-ATP-Competitive Protein Kinase Inhibitors for Oncology

被引：8
|
作者：
McInnes, Campbell [1 ]
机构：
[1] Univ S Carolina, S Carolina Coll Pharm, Columbia, SC 29208 USA
来源：
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 47 | 2012年 / 47卷
关键词：
POLO-LIKE KINASE-1; BOX DOMAIN; DNA-DAMAGE; PEPTIDE INHIBITORS; RECRUITMENT-SITE; DESIGN; PHOSPHORYLATION; IDENTIFICATION; COMPLEX; POLO-LIKE-KINASE-1;
D O I：
10.1016/B978-0-12-396492-2.00029-1
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：459 / 474
页数：16
相关论文
共 50 条
  • [1] Identification of non-ATP-competitive α-carboline inhibitors of the anaplastic lymphoma kinase
    Mologni, Luca
    Orsato, Alexandre
    Zambon, Alfonso
    Tardy, Sebastien
    Bisson, William H.
    Schneider, Cedric
    Ceccon, Monica
    Viltadi, Michela
    D'Attoma, Joseph
    Pannilunghi, Sara
    Vece, Vito
    Gueyrard, David
    Bertho, Jerome
    Scapozza, Leonardo
    Goekjian, Peter
    Gambacorti-Passerini, Carlo
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 238
  • [2] Non-ATP-competitive kinase inhibitors - enhancing selectivity through new inhibition strategies
    Harrison, Stephen
    Das, Kanad
    Karim, Felix
    Maclean, Derek
    Mendel, Dirk
    EXPERT OPINION ON DRUG DISCOVERY, 2008, 3 (07) : 761 - 774
  • [3] Serotonin derivatives as a new class of non-ATP-competitive receptor tyrosine kinase inhibitors
    Buettner, Anita
    Cottin, Thomas
    Xu, Jing
    Tzagkaroulaki, Lito
    Giannis, Athanassios
    BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 18 (10) : 3387 - 3402
  • [4] Discovery of Non-ATP-Competitive Inhibitors of Polo-like Kinase1
    Yun, Taikangxiang
    Qin, Tan
    Liu, Ying
    Lai, Luhua
    CHEMMEDCHEM, 2016, 11 (07) : 713 - 717
  • [5] Non-ATP Competitive Protein Kinase Inhibitors
    Garuti, L.
    Roberti, M.
    Bottegoni, G.
    CURRENT MEDICINAL CHEMISTRY, 2010, 17 (25) : 2804 - 2821
  • [6] Development of Selective Phosphatidylinositol 5-Phosphate 4-Kinase γ Inhibitors with a Non-ATP-competitive, Allosteric Binding Mode
    Boffey, Helen K.
    Rooney, Timothy P. C.
    Willems, Henriette M. G.
    Edwards, Simon
    Green, Christopher
    Howard, Tina
    Ogg, Derek
    Romero, Tamara
    Scott, Duncan E.
    Winpenny, David
    Duce, James
    Skidmore, John
    Clarke, Jonathan H.
    Andrews, Stephen P.
    JOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (04) : 3359 - 3370
  • [7] Recent progress in the development of ATP-Competitive and allosteric akt kinase inhibitors
    Lindsley, Craig W.
    Barnett, Stanley F.
    Yaroschak, Melissa
    Bilodeau, Mark T.
    Layton, Mark E.
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2007, 7 (14) : 1349 - 1363
  • [8] A biochemical approach to discriminate between ATP-competitive and non-ATP competitive protein kinase inhibitors
    Mueller, Daniel
    Totzke, Frank
    Weber, Thomas
    Heidemann-Dinger, Carolin
    Ketterer, Constance
    Kramer, Diane
    Pathe, Marcel
    Kubbutat, Michael H.
    CANCER RESEARCH, 2017, 77
  • [9] Recent progress in development of non-ATP competitive small-molecule inhibitors of protein kinases
    Kiselyov, Alex
    Balakin, Konstantin V.
    Tkachenko, Sergey E.
    Savchuk, Nikolay P.
    MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2006, 6 (06) : 711 - 717
  • [10] Experimental non-ATP-competitive therapies for chronic myelogenous leukemia
    A Quintás-Cardama
    Leukemia, 2008, 22 : 932 - 940
12345