Binding of [H-3]-terazosin and its enantiomers at alpha(1)-adrenoceptor subtypes

被引:0
|
作者
Ireland, LM [1 ]
Rotert, G [1 ]
Shoghi, S [1 ]
Thomas, S [1 ]
Cain, JC [1 ]
Hancock, AA [1 ]
Kerwin, JF [1 ]
机构
[1] ABBOTT LABS,ABBOTT PK,IL 60064
来源
FASEB JOURNAL | 1996年 / 10卷 / 03期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:2415 / 2415
页数:1
相关论文
共 50 条
  • [31] COMPARISON OF BOVINE PLATELET AND TEAT ALPHA-2-ADRENOCEPTOR CHARACTERISTICS BY [H-3] RAUWOLSCINE BINDING
    ROETS, E
    BURVENICH, C
    PEETERS, G
    ARCHIVES INTERNATIONALES DE PHARMACODYNAMIE ET DE THERAPIE, 1988, 293 : 175 - 185
  • [32] Tamsulosin:: Assessment of affinity of 3H-prazosin binding to two alpha-1-adrenoceptor subtypes in the canine aorta
    Nakamura, T
    Maruyama, K
    Ohnuki, T
    Hattori, K
    Watanabe, K
    Nagatomo, T
    PHARMACOLOGY, 1999, 59 (05) : 234 - 238
  • [33] CLASSIFICATION OF ALPHA(1)-ADRENOCEPTOR SUBTYPES
    MICHEL, MC
    KENNY, B
    SCHWINN, DA
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1995, 352 (01) : 1 - 10
  • [34] HETEROGENEOUS H-3 RAUWOLSCINE BINDING-SITES IN RAT CORTEX - 2 ALPHA-2-ADRENOCEPTOR SUBTYPES OR AN ADDITIONAL NON-ADRENERGIC INTERACTION
    BROADHURST, AM
    ALEXANDER, BS
    WOOD, MD
    LIFE SCIENCES, 1988, 43 (01) : 83 - 92
  • [35] CHARACTERIZATION OF ALPHA-ADRENERGIC RECEPTOR SUBTYPES IN RAT-BRAIN BY BINDING OF [H-3]-DIHYDROERGOCRYPTINE
    HAGA, T
    HAGA, K
    NEUROCHEMICAL RESEARCH, 1981, 6 (01) : 101 - 101
  • [36] CHARACTERIZATION OF [H-3] RX821002 BINDING TO ALPHA-2-ADRENERGIC RECEPTOR SUBTYPES
    OROURKE, MF
    BLAXALL, HS
    IVERSEN, LJ
    BYLUND, DB
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1994, 268 (03): : 1362 - 1367
  • [37] Non-adrenoceptor binding of [H-3]atipamezole in rat kidney
    Sjoholm, B
    Lahdesmaki, J
    Scheinin, M
    BRITISH JOURNAL OF PHARMACOLOGY, 1996, 119 : P322 - P322
  • [38] PHARMACOLOGICAL EVIDENCE FOR ALPHA-2 ADRENOCEPTOR HETEROGENEITY - DIFFERENTIAL BINDING-PROPERTIES OF [H-3] RAUWOLSCINE AND [H-3] IDAZOXAN IN RAT-BRAIN
    BOYAJIAN, CL
    LESLIE, FM
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1987, 241 (03): : 1092 - 1098
  • [39] [H-3] MK-912 BINDING DELINEATES 2 ALPHA-2-ADRENOCEPTOR SUBTYPES IN RAT CNS ONE OF WHICH IS IDENTICAL WITH THE CLONED PA2D ALPHA-2-ADRENOCEPTOR
    UHLEN, S
    XIA, Y
    CHHAJLANI, V
    FELDER, CC
    WIKBERG, JES
    BRITISH JOURNAL OF PHARMACOLOGY, 1992, 106 (04) : 986 - 995
  • [40] 2 DISTINCT ALPHA(1)-ADRENOCEPTOR SUBTYPES IN RABBIT LIVER - A BINDING STUDY
    OHMURA, T
    MURAMATSU, I
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 116 (06) : 2591 - 2596