Annelated Pyrrolo[1,2-a][1,4]diazepines in Mannich Reaction

被引：2
|
作者：
Stroganova, Tatyana A. [1 ]
Red'kin, Viktor M. [1 ]
Vasilin, Vladimir K. [1 ]
Krapivin, Gennady D. [1 ]
机构：
[1] Kuban State Technol Univ, Krasnodar 350072, Russia
来源：
JOURNAL OF HETEROCYCLIC CHEMISTRY | 2013年 / 50卷 / 04期
关键词：
BETA-AMINOMETHYLATION; BASES; ANTIFUNGAL; PYRROLES; AGENTS;
D O I：
10.1002/jhet.1581
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New Mannich bases were synthesized through an interaction of fused pyrrolo[1,2-a][1,4]diazepines with secondary amines and formaldehyde. The reaction appears to be regioselective, yielding the monosubstituted products bearing N,N-dialkylaminomethyl group at position 2 of the pyrrolodiazepine moiety.
引用
收藏
页码：854 / 858
页数：5
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