Annelated Pyrrolo[1,2-a][1,4]diazepines in Mannich Reaction

被引：2

作者：

Stroganova, Tatyana A. ^{[1
]}

Red'kin, Viktor M. ^{[1
]}

Vasilin, Vladimir K. ^{[1
]}

Krapivin, Gennady D. ^{[1
]}

机构：

[1] Kuban State Technol Univ, Krasnodar 350072, Russia

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2013年 / 50卷 / 04期

关键词：

BETA-AMINOMETHYLATION; BASES; ANTIFUNGAL; PYRROLES; AGENTS;

D O I：

10.1002/jhet.1581

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

New Mannich bases were synthesized through an interaction of fused pyrrolo[1,2-a][1,4]diazepines with secondary amines and formaldehyde. The reaction appears to be regioselective, yielding the monosubstituted products bearing N,N-dialkylaminomethyl group at position 2 of the pyrrolodiazepine moiety.

引用

页码：854 / 858

页数：5

共 50 条

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