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- [2] Seletalisib: Characterization of a Novel, Potent, and Selective Inhibitor of PI3KδJOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2017, 361 (03): : 429 - 440Allen, Rodger A.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandBrookings, Daniel C.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandPowell, Mark J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Immunocore Ltd, Abingdon, Oxon, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandDelgado, Jean论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandShuttleworth, Lindsay K.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandMerriman, Mark论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandFahy, Ian J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Beckman Coulter, High Wycombe, Bucks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandTewari, Roohi论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandSilva, John P.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandHealy, Louise J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Aurelia Biosci, Nottingham, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandDavies, Gareth C. G.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandTwomey, Breda论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandCutler, Rona M.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandKotian, Apoorva论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandCrosby, Andrea论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandMcCluskey, Gillian论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandWatt, Gillian F.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandPayne, Andrew论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England
- [3] Dual PI3K/ERK inhibitor AEZS-136, a potent antitumor compound under preclinical developmentABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 244Gerlach, Matthias论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanySeipelt, Irene论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyBlumenstein, Lars论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyJung, Kai论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanySchuster, Tilmann论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyMueller, Gilbert论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyGuenther, Eckhard论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyEngel, Juergen论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, GermanyTeifel, Michael论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany Aeterna Zentaris GmbH, D-60314 Frankfurt, Hesse, Germany
- [4] Discovery of a novel and potent mutant-selective inhibitor of PI3KαCANCER RESEARCH, 2024, 84 (06)Gao, Mingming论文数: 0 引用数: 0 h-index: 0Qi, Chao论文数: 0 引用数: 0 h-index: 0Li, Zhentian论文数: 0 引用数: 0 h-index: 0Fan, Qipeng论文数: 0 引用数: 0 h-index: 0Wang, Liyang论文数: 0 引用数: 0 h-index: 0Zhou, Fei论文数: 0 引用数: 0 h-index: 0You, Lin论文数: 0 引用数: 0 h-index: 0Zheng, Hewen论文数: 0 引用数: 0 h-index: 0Li, Yu论文数: 0 引用数: 0 h-index: 0Wu, Liangxing论文数: 0 引用数: 0 h-index: 0Yao, Wenqing论文数: 0 引用数: 0 h-index: 0Liu, Phillip C.论文数: 0 引用数: 0 h-index: 0
- [5] Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitorBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (14) : 3917 - 3924Hamajima, Toshihiro论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanTakahashi, Fumie论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKato, Koji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanSugano, Yukihito论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYamaki, Susumu论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanMoritomo, Ayako论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanKubo, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanNakamura, Koji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYamagami, Kaoru论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanHamakawa, Nozomu论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanYokoo, Koji论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, JapanFukahori, Hidehiko论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan Astellas Pharma Inc, Drug Discovery Res, 21 Miyukigaoka, Tsukuba, Ibaraki 3058585, Japan
- [6] In vitro characterization of AMG 511, a potent and selective class I PI3K inhibitor for the treatment of cancerCANCER RESEARCH, 2012, 72Caenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAZhang, Nancy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAWang, Ling论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USANorman, Mark H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USABurgess, Terri论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USARadinsky, Robert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKendall, Rick论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAFreeman, Daniel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAHughes, Paul E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USA
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