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- [1] AMG 511, a potent and selective class I PI3K inhibitor, suppresses the growth of Kras mutant lung tumors in mice[J]. CANCER RESEARCH, 2012, 72Estrada, Juan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAUngersma, Sharon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKaufman, Stephen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAYerby, Brittany论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAZhang, Nancy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAFreeman, Daniel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAHughes, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USASilva, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USACoxon, Angela论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USA
- [2] AMG 511, a potent and selective class I PI3K inhibitor, demonstrates anti-tumor activity in multiple xenograft models[J]. CANCER RESEARCH, 2012, 72Zhang, Nancy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USACaenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAWang, Ling论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USANorman, Mark论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKendall, Richard论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USABurgess, Terri论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USARadinsky, Robert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAHughes, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAFreeman, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USA
- [3] Seletalisib: Characterization of a Novel, Potent, and Selective Inhibitor of PI3Kδ[J]. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2017, 361 (03): : 429 - 440Allen, Rodger A.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandBrookings, Daniel C.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandPowell, Mark J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Immunocore Ltd, Abingdon, Oxon, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandDelgado, Jean论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandShuttleworth, Lindsay K.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandMerriman, Mark论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandFahy, Ian J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Beckman Coulter, High Wycombe, Bucks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandTewari, Roohi论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandSilva, John P.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandHealy, Louise J.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England Aurelia Biosci, Nottingham, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandDavies, Gareth C. G.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandTwomey, Breda论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandCutler, Rona M.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandKotian, Apoorva论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandCrosby, Andrea论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandMcCluskey, Gillian论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandWatt, Gillian F.论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, EnglandPayne, Andrew论文数: 0 引用数: 0 h-index: 0机构: UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England UCB Pharma Ltd, 216 Bath Rd, Slough SL1 4EN, Berks, England
- [4] A novel, highly potent PI3Kα covalent inhibitor deconvolutes class I PI3K isoforms in cancer cells.[J]. CANCER RESEARCH, 2021, 81 (13)Keles, Erhan论文数: 0 引用数: 0 h-index: 0机构: Univ Basel, Basel, Switzerland Univ Basel, Basel, Switzerland论文数: 引用数: h-index:机构:Sriramaratnam, Rohitha论文数: 0 引用数: 0 h-index: 0机构: Univ Basel, Basel, Switzerland Univ Basel, Basel, SwitzerlandSchafer, Thorsten论文数: 0 引用数: 0 h-index: 0机构: Univ Basel, Basel, Switzerland Univ Basel, Basel, SwitzerlandWymann, Matthias P.论文数: 0 引用数: 0 h-index: 0机构: Univ Basel, Basel, Switzerland Univ Basel, Basel, Switzerland
- [5] Identification of AMG 511 as a selective class I phosphoinositide 3-kinase inhibitor[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245Wurz, Ryan P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAAndrews, Kristin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Mol Struct, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USABo, Yunxin Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USABooker, Shon K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USACaenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USACee, Victor J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USANoel, D'Angelo D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAFreeman, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAHerberich, Bradley J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAHong, Fang-Tsao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAJackson, Claire L. M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAJiang, Jian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USALanman, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USALiu, Longbin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAMcCarter, John D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, High Throughput Screening Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAMullady, Erin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, High Throughput Screening Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USANishimura, Nobuko论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAPettus, Liping H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAReed, Anthony B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USASan Miguel, Tisha论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, High Throughput Screening Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USASmith, Adrian L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAStec, Markian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USATadesse, Seifu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USATasker, Andrew S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAAidasani, Divesh论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAZhu, Xiaochun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USASubramanian, Raju论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USATamayo, Nuria A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAWang, Ling论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAWhittington, Douglas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAWu, Bin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAWu, Tian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmaceut, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAYang, Kevin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAZalameda, Leeanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, High Throughput Screening Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAZhang, Nancy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USAHughes, Paul E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USANorman, Mark H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Med Chem, Thousand Oaks, CA 91320 USA
- [6] In vitro profiling of the potent and selective PI3K inhibitor AEZS-126[J]. CANCER RESEARCH, 2009, 69Seipelt, Irene论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyGerlach, Matthias论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyBlumenstein, Lars论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyMueller, Gilbert论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyTeifel, Michael论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyPolymeropoulos, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, GermanyGuenther, Eckhard论文数: 0 引用数: 0 h-index: 0机构: Aeterna Zentaris GmbH, Frankfurt, Germany Aeterna Zentaris GmbH, Frankfurt, Germany
- [7] INK1117: A potent and orally efficacious PI3Kα-selective inhibitor for the treatment of cancer[J]. CANCER RESEARCH, 2011, 71Jessen, Katayoun A.论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAKessler, Linda论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAKucharski, Jeff论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAGuo, Xin论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAStaunton, Jocelyn论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAElia, Marikka论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAJanes, Matthew论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USALan, Lucy论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAWang, Shunyou论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAStewart, Josh论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USADarjania, Levan论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USALi, Liansheng论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAChan, Katrina论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAMartin, Michael论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USARen, Pingda论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USAFruman, David论文数: 0 引用数: 0 h-index: 0机构: UC Irvine, Irvine, CA USA Intellikine, La Jolla, CA USARommel, Christian论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USALiu, Yi论文数: 0 引用数: 0 h-index: 0机构: Intellikine, La Jolla, CA USA Intellikine, La Jolla, CA USA
- [8] Discovery of a Potent, Selective, and Orally Available PI3Kδ Inhibitor for the Treatment of Inflammatory Diseases[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2017, 8 (01): : 118 - 123Erra, Montse论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainTaltavull, Joan论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainGreco, Angelique论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Pharmaxis Ltd, 20 Rodborough Rd, Frenchs Forest, NSW 2086, Australia Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainJavier Bernal, Francisco论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainFrancisco Caturla, Juan论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainGracia, Jordi论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainDominguez, Maria论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Pharmacokinet & Metab, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainSabate, Mar论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Pharmacokinet & Metab, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainParis, Stephane论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainSoria, Salome论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainHernandez, Begona论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain Fundacio ACE, Marques Sentmenat,57, Barcelona 08029, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainArmengol, Clara论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainCabedo, Judit论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Syst Biol, Barcelona 08980, Spain Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainBravo, Monica论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainCalama, Elena论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainMiralpeix, Montserrat论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Almirall R&D, Med Chem & Screening, Barcelona 08980, SpainLehner, Martin D.论文数: 0 引用数: 0 h-index: 0机构: Almirall R&D, Resp Therapeut Area, Barcelona 08980, Spain Bionor SE, Kerschensteinerstr 11-15, D-92318 Neumarkt, Germany Almirall R&D, Med Chem & Screening, Barcelona 08980, Spain
- [9] Characterization of a potent inhibitor of class 1 phosphatidylinositide-3′-kinases (PI3K) in human glioma[J]. MOLECULAR CANCER THERAPEUTICS, 2007, 6 (12) : 3414S - 3414SClarke, Paul A.论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandGuillard, Sandrine论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandDi Stefano, Francesca论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandPoele, Robert te论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandValenti, Melanie论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandBrandon, Alexis de Haven论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandEccles, Sue论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandRaynaud, Florence论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, EnglandWorkman, Paul论文数: 0 引用数: 0 h-index: 0机构: CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England CR UK Ctr Canc Therapeut, Inst Canc Res, Sutton, Surrey, England
- [10] Discovery of a novel and potent mutant-selective inhibitor of PI3Kα[J]. CANCER RESEARCH, 2024, 84 (06)Gao, Mingming论文数: 0 引用数: 0 h-index: 0Qi, Chao论文数: 0 引用数: 0 h-index: 0Li, Zhentian论文数: 0 引用数: 0 h-index: 0Fan, Qipeng论文数: 0 引用数: 0 h-index: 0Wang, Liyang论文数: 0 引用数: 0 h-index: 0Zhou, Fei论文数: 0 引用数: 0 h-index: 0You, Lin论文数: 0 引用数: 0 h-index: 0Zheng, Hewen论文数: 0 引用数: 0 h-index: 0Li, Yu论文数: 0 引用数: 0 h-index: 0Wu, Liangxing论文数: 0 引用数: 0 h-index: 0Yao, Wenqing论文数: 0 引用数: 0 h-index: 0Liu, Phillip C.论文数: 0 引用数: 0 h-index: 0