Design and optimization of benzimidazole-containing cold menthol receptor (TRPM8) antagonists

被引:0
|
作者
Parks, Daniel J. [1 ]
Calvo, Raul R. [1 ]
Parsons, William H. [1 ]
Meegalla, Sanath [1 ]
Ballentine, Shelley K. [1 ]
Chen, Jinsheng [1 ]
Illig, Carl R. [1 ]
Stone, Dennis J. [1 ]
Qin, Ning [1 ]
Hutchinson, Tasha L. [1 ]
Lubin, Mary Lou [1 ]
Liu, Yi [1 ]
Baker, Judith [1 ]
Colburn, Raymond W. [1 ]
Flores, Christopher M. [1 ]
Player, Mark R. [1 ]
机构
[1] Johnson & Johnson Pharmaceut Res & Dev, Spring House, PA USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
425-MEDI
引用
收藏
页数:1
相关论文
共 50 条
  • [31] THE EFFECTS OF VARIATIONS IN THE N-TERMINUS ON THE SENSITIVITY OF CHICK TRPM8 TO MENTHOL AND COLD
    Morshed, N.
    Reid, G.
    IRISH JOURNAL OF MEDICAL SCIENCE, 2011, 180 : S297 - S298
  • [32] Effects of Antagonists and Heat on TRPM8 Channel Currents in Dorsal Root Ganglion Neuron Activated by Nociceptive Cold Stress and Menthol
    Mustafa Nazıroğlu
    Cemil Özgül
    Neurochemical Research, 2012, 37 : 314 - 320
  • [33] Effects of Antagonists and Heat on TRPM8 Channel Currents in Dorsal Root Ganglion Neuron Activated by Nociceptive Cold Stress and Menthol
    Naziroglu, Mustafa
    Ozgul, Cemil
    NEUROCHEMICAL RESEARCH, 2012, 37 (02) : 314 - 320
  • [34] Optical Control of TRPM8 Channels with Photoswitchable Menthol
    Becker, Jasmin
    Ellerkmann, Clara S.
    Schmelzer, Hannah
    Hermann, Christian
    Lützel, Kyra
    Gudermann, Thomas
    Konrad, David B.
    Trauner, Dirk
    Storch, Ursula
    Mederos y Schnitzler, Michael
    Angewandte Chemie - International Edition, 2025, 64 (05)
  • [35] Opiates Modulate Thermosensation by Internalizing Cold Receptor TRPM8
    Shapovalov, George
    Gkika, Dimitra
    Devilliers, Maily
    Kondratskyi, Artem
    Gordienko, Dmitri
    Busserolles, Jerome
    Bokhobza, Alexandre
    Eschalier, Alain
    Skryma, Roman
    Prevarskaya, Natalia
    CELL REPORTS, 2013, 4 (03): : 504 - 515
  • [36] TRPM8 and prostate: a cold case?
    Noyer, Lucile
    Grolez, Guillaume P.
    Prevarskaya, Natalia
    Gkika, Dimitra
    Lemonnier, Loic
    PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 2018, 470 (10): : 1419 - 1429
  • [37] Cool and menthol receptor TRPM8 in human urinary bladder disorders and clinical correlations
    Mukerji G.
    Yiangou Y.
    Corcoran S.L.
    Selmer I.S.
    Smith G.D.
    Benham C.D.
    Bountra C.
    Agarwal S.K.
    Anand P.
    BMC Urology, 6 (1)
  • [38] TRPM8 and prostate: a cold case?
    Lucile Noyer
    Guillaume P. Grolez
    Natalia Prevarskaya
    Dimitra Gkika
    Loic Lemonnier
    Pflügers Archiv - European Journal of Physiology, 2018, 470 : 1419 - 1429
  • [39] Arylglycine derivatives as potent antagonists of transient receptor potential melastatin 8 (TRPM8)
    Zhu, Bin
    Xia, Mingde
    Xu, Xiaoqing
    Ludovici, Donald W.
    Tennakoon, Manomi
    Youngman, Mark A.
    Matthews, Jay M.
    Dax, Scott L.
    Colburn, Raymond W.
    Qin, Ning
    Hutchinson, Tasha L.
    Lubin, Mary Lou
    Brandt, Michael R.
    Stone, Dennis J.
    Flores, Christopher M.
    Macielag, Mark J.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 244
  • [40] Arylglycine derivatives as potent transient receptor potential melastatin 8 (TRPM8) antagonists
    Zhu, Bin
    Xia, Mingde
    Xu, Xiaoqing
    Ludovici, Donald W.
    Tennakoon, Manomi
    Youngman, Mark A.
    Matthews, Jay M.
    Dax, Scott L.
    Colburn, Raymond W.
    Qin, Ning
    Hutchinson, Tasha L.
    Lubin, Mary Lou
    Brandt, Michael R.
    Stone, Dennis J.
    Flores, Christopher M.
    Macielag, Mark J.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (07) : 2234 - 2237