Synthesis and antimicrobial screening of novel 2,6-ditertiarybutylpiperidin-4-ones

被引：1

作者：

Govindaraju, C. ^{[1
]}

Valliappan, R. ^{[2
]}

Sundari, V. ^{[3
]}

机构：

[1] Annamalai Univ, Dept Chem, Annamalainagar 608002, Tamil Nadu, India

[2] Annamalai Univ, DDE, Annamalainagar 608002, Tamil Nadu, India

[3] Annamalai Univ, FEAT, Annamalainagar 608002, Tamil Nadu, India

来源：

MEDICINAL CHEMISTRY RESEARCH | 2012年 / 21卷 / 11期

关键词：

Trimethylacetaldehyde; 2,6-Ditertiarybutylpiperidine-4-one; Antibacterial; Antifungal;

D O I：

10.1007/s00044-011-9913-9

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A new series of 2,6-ditertiarybutyl 4-piperidones were prepared from an aliphatic aldehyde not having an alpha hydrogen atom and their structures were confirmed by elemental and spectral data. These compounds were screened for antibacterial (Bacillus subtilis, Escherichia coli, and Klebsiella pneumonia) and antifungal (Aspergillus niger and Trichoderma sp.) activities and found to be potentially active against bacteria and fungi.

引用

页码：3687 / 3691

页数：5

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