Facile and convenient synthesis of pyrazole, pyridine, pyridazine, pyrazolo[3,4-b]pyridine, and pyrazolo[5,1-c][1,2,4]triazine derivatives

被引：23

作者：

Kheder, Nabila A. ^{[1
]}

Mabkhot, Yahia N. ^{[2
]}

Farag, Ahmad M. ^{[1
]}

机构：

[1] Cairo Univ, Dept Chem, Fac Sci, Giza 12613, Egypt

[2] Zamar Univ, Fac Sci, Dept Chem, Zamar, Yemen

来源：

SYNTHETIC COMMUNICATIONS | 2008年 / 38卷 / 18期

关键词：

N-(pyrimid-2-yl) butanamide; imidazo[1,2-a] pyrimidine; pyrazole; pyrazolo[3,4-b] pyridine; pyrazolo[5,1-c][1,2,4] triazine; pyridazine; pyridinethione;

D O I：

10.1080/00397910802109257

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A convenient synthesis of a series of pyrazole, pyridine, pyridinethione, pyridazine, pyrazolo[3,4-b]pyridine, imidazo[1,2-a]pyrimidine, and pyrazolo[5,1-c][1, 2, 4]triazine derivatives incorporating a pyrimidine moiety, via the reactions of the versatile, readily accessible 3-oxo-N-(pyrimid-2-yl)butanamide with the appropriate reagents, is described.

引用

页码：3170 / 3182

页数：13

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