DEVELOPMENT OF A HIGH-THROUGHPUT IN-VITRO SCREEN TO IDENTIFY INHIBITORS OF THE PLASMODIUM FALCIPARUM HEAT SHOCK PROTEIN 90 BINDING ACTIVITY

被引：0
|
作者：
Kramer, Martin L. [1 ]
Patel, Vishal [2 ]
Clardy, Jon [2 ]
Wirth, Dyann F. [3 ]
机构：
[1] Genzyme Corp, Waltham, MA USA
[2] Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA
[3] Harvard Univ, Sch Publ Hlth, Dept Immunol & Infect Dis, Boston, MA 02115 USA
来源：
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE | 2008年 / 79卷 / 06期
关键词：
D O I：
暂无
中图分类号：
R1 [预防医学、卫生学];
学科分类号：
1004 ; 120402 ;
摘要：
588
引用
收藏
页码：174 / 174
页数：1
相关论文
共 50 条
  • [41] Yeast-Based High-Throughput Screen Identifies Plasmodium falciparum Equilibrative Nucleoside Transporter 1 Inhibitors That Kill Malaria Parasites
    Frame, I. J.
    Deniskin, Roman
    Rinderspacher, Alison
    Katz, Francine
    Deng, Shi-Xian
    Moir, Robyn D.
    Adjalley, Sophie H.
    Coburn-Flynn, Olivia
    Fidock, David A.
    Willis, Ian M.
    Landry, Donald W.
    Akabas, Myles H.
    ACS CHEMICAL BIOLOGY, 2015, 10 (03) : 775 - 783
  • [42] Plasmodium falciparum Heat Shock Protein 70 Lacks Immune Modulatory Activity
    Pooe, Ofentse Jacob
    Koellisch, Gabriele
    Heine, Holger
    Shonhai, Addmore
    PROTEIN AND PEPTIDE LETTERS, 2017, 24 (06): : 503 - 510
  • [43] Development of a High-Throughput Assay to Identify Inhibitors of ENPP1
    Kumar, Meera
    Lowery, Robert G.
    SLAS DISCOVERY, 2021, 26 (05) : 740 - 746
  • [44] IN-VITRO ACTIVITY OF MITOCHONDRIAL ATP-SYNTHETASE INHIBITORS AGAINST PLASMODIUM-FALCIPARUM
    BASCO, LK
    LEBRAS, J
    JOURNAL OF EUKARYOTIC MICROBIOLOGY, 1994, 41 (03) : 179 - 183
  • [45] Development of a high-throughput in vitro assay to identify selective inhibitors for human ALDH1A1
    Morgan, Cynthia A.
    Hurley, Thomas D.
    CHEMICO-BIOLOGICAL INTERACTIONS, 2015, 234 : 29 - 37
  • [46] Plasmodium falciparum calcineurin and its association with heat shock protein 90:: mechanisms for the antimalarial activity of cyclosporin A and synergism with geldanamycin
    Kumar, R
    Musiyenko, A
    Barik, S
    MOLECULAR AND BIOCHEMICAL PARASITOLOGY, 2005, 141 (01) : 29 - 37
  • [47] The heat shock protein 90 of Plasmodium falciparum and antimalarial activity of its inhibitor, geldanamycin -: art. no. 30
    Kumar, R
    Musiyenko, A
    Barik, S
    MALARIA JOURNAL, 2003, 2 (1)
  • [48] Development of a high-throughput screen for inhibitors of replication protein A and its role in DNA replication and repair.
    Turchi, JJ
    Andrews, BJ
    CLINICAL CANCER RESEARCH, 2003, 9 (16) : 6175S - 6175S
  • [49] A High-Throughput Screen for Receptor Protein Tyrosine Phosphatase-γ Selective Inhibitors
    Appiah, Kingsley K.
    Kostich, Walter A.
    Gerritz, Samuel W.
    Huang, Yanling
    Hamman, Brian D.
    Allen, Jason
    Zhang, Wandong
    Lanthorn, Thomas H.
    Albright, Charles F.
    Westphal, Ryan
    Banks, Martyn N.
    O'Connell, Jonathan C.
    JOURNAL OF BIOMOLECULAR SCREENING, 2011, 16 (05) : 476 - 485
  • [50] A High-Throughput Screen To Identify Inhibitors of ATP Homeostasis in Non-replicating Mycobacterium tuberculosis
    Mak, Puiying A.
    Rao, Srinivasa P. S.
    Tan, Mai Ping
    Lin, Xiuhua
    Chyba, Jason
    Tay, Joann
    Ng, Seow Hwee
    Tan, Bee Huat
    Cherian, Joseph
    Duraiswamy, Jeyaraj
    Bifani, Pablo
    Lim, Vivian
    Lee, Boon Heng
    Ma, Ngai Ling
    Beer, David
    Thayalan, Pamela
    Kuhen, Kelli
    Chatterjee, Arnab
    Supek, Frantisek
    Glynne, Richard
    Zheng, Jun
    Boshoff, Helena I.
    Barry, Clifton E., III
    Dick, Thomas
    Pethe, Kevin
    Camacho, Luis R.
    ACS CHEMICAL BIOLOGY, 2012, 7 (07) : 1190 - 1197
12345