Synthesis, Structure and Biological Activities of 2,2-Dichloro-1-(4-ethoxyphenyl)-cyclopropanyl Substituted Piperidin-1-yl Ketone

被引：6
|
作者：
Sun, Na-Bo [1 ]
Jin, Jian-Zhong [1 ]
Lei, Chao [1 ]
Ke, Wei [1 ]
机构：
[1] Zhejiang Shuren Univ, Coll Biol & Environm Engn, Hangzhou 310015, Zhejiang, Peoples R China
来源：
ASIAN JOURNAL OF CHEMISTRY | 2013年 / 25卷 / 07期
关键词：
Pyrethroid; Cycloprothrin; Piperidine; Synthesis; Structure; CRYSTAL-STRUCTURE; CYCLOPROPANE MOIETY; DFT CALCULATION; ANTIFUNGAL ACTIVITY; DERIVATIVES; BIOACTIVITY;
D O I：
10.14233/ajchem.2013.14040
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Ten new amide-type compounds, which are pyrethroids containing piperidine, are synthesized from 1-(4-ethyoxyphenyl)-2,2-dichlorocyclopropane-1-carboxylic acid and substituted piperidine. Their structures were confirmed by H-1 NMR, MS and elemental analysis. The crystal structure of 4a and 4h were determined by X-ray diffraction analysis. The bioassay results indicated that they showed moderate activity.
引用
收藏
页码：4067 / 4070
页数：4
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