Synthesis and biological evaluation of clitocine analogs as adenosine kinase inhibitors.

被引：0
|
作者：
Lee, CH [1 ]
Jiang, MQ [1 ]
Daanen, J [1 ]
Kohlaas, KL [1 ]
Alexander, KM [1 ]
Yu, HX [1 ]
Kowaluk, EA [1 ]
Bhagwat, SS [1 ]
机构：
[1] ABBOTT LABS,NEUROSCI RES,ABBOTT PK,IL 60064
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 1996年 / 212卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：156 / MEDI
页数：1
相关论文
共 50 条
  • [41] Synthesis and biological evaluation of BIRB 796 analogs as potent inhibitors of p38 MAP kinase.
    Swinamer, AD
    Capolino, A
    Cirillo, PF
    Gilmore, T
    Graham, A
    Hickey, E
    Moriak, M
    Madwed, J
    Moss, N
    Nelson, R
    Pargellis, C
    Regan, J
    Torcellini, C
    Tsang, M
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U59 - U60
  • [42] Synthesis and biological evaluation of 2-epi-jaspine B analogs as selective sphingosine kinase 1 inhibitors
    Yang, Haoran
    Li, Ying
    Chai, Huining
    Yakura, Takayuki
    Liu, Bo
    Yao, Qingqiang
    BIOORGANIC CHEMISTRY, 2020, 98
  • [43] SYNTHESIS AND BIOLOGICAL EVALUATION OF CONFORMATIONALLY CONSTRAINED BICYCLIC AND TRICYCLIC BALANOL ANALOGS AS INHIBITORS OF PROTEIN-KINASE-C
    MENDOZA, JS
    JAGDMANN, GE
    GOSNELL, PA
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (19) : 2211 - 2216
  • [44] Design, synthesis, and SAR of 6-alkynylpyrimidines as potent, selective, and in vivo active adenosine kinase inhibitors.
    Gomtsyan, A
    Didomenico, S
    Lee, CH
    Matulenko, M
    Stewart, A
    Kowaluk, E
    Wismer, C
    Mikusa, J
    Yu, HX
    Kohlhaas, K
    Jarvis, M
    Bhagwat, S
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 222 : U679 - U679
  • [45] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CARBOCYCLIC CLITOCINE
    BAXTER, AD
    PENN, CR
    STORER, R
    WEIR, NG
    WOODS, JM
    NUCLEOSIDES & NUCLEOTIDES, 1991, 10 (1-3): : 393 - 396
  • [46] ROLE OF ADENOSINE KINASE IN THE BIOLOGICAL (ANTIVIRAL AND ANTICELLULAR) ACTIVITIES OF ADENOSINE-ANALOGS
    COOLS, M
    DECLERCQ, E
    DRACH, JC
    NUCLEOSIDES & NUCLEOTIDES, 1987, 6 (1-2): : 423 - 424
  • [47] Synthesis and biological evaluation of naphthoquinone analogs as a novel class of proteasome inhibitors
    Lawrence, Harshani R.
    Kazi, Aslamuzzaman
    Luo, Yunting
    Kendig, Robert
    Ge, Yiyu
    Jain, Sanjula
    Daniel, Kenyon
    Santiago, Daniel
    Guida, Wayne C.
    Sebti, Said M.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 18 (15) : 5576 - 5592
  • [48] Synthesis and Biological Evaluation of Ezetimibe Analogs as Possible Cholesterol Absorption Inhibitors
    Wang, Yubin
    Haiqian
    Huang, Wenlong
    Zhang, Huibin
    Zhou, Jinpei
    LETTERS IN DRUG DESIGN & DISCOVERY, 2011, 8 (06) : 500 - 505
  • [49] Myxopyronin B analogs as inhibitors of RNA polymerase, synthesis and biological evaluation
    Doundoulakis, T
    Xiang, AX
    Lira, R
    Agrios, KA
    Webber, SE
    Sisson, W
    Aust, RM
    Shah, AM
    Showalter, RE
    Appleman, JR
    Simonsen, KB
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (22) : 5667 - 5672
  • [50] Synthesis, biological evaluation, and docking studies of gigantol analogs as calmodulin inhibitors
    Reyes-Ramirez, Adelfo
    Leyte-Lugo, Martha
    Figueroa, Mario
    Serrano-Alba, Trinidad
    Gonzalez-Andrade, Martin
    Mata, Rachel
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 46 (07) : 2699 - 2708
12345