Radiosynthesis and in vitro evaluation of a series of novel homologous [18F]-labeled dopamine D2/3-agonist ligands

被引：0
|
作者：
Shalgunov, Vladimir [1 ]
Dierckx, Rudi A. J. O. [1 ]
Janssen, Henk M. [2 ]
Booij, Jan [3 ]
Elsinga, Philip H. [1 ]
机构：
[1] Univ Groningen, Univ Med Ctr Groningen, NL-9700 AB Groningen, Netherlands
[2] SyMO Chem BV, TU E, Eindhoven, Netherlands
[3] Univ Amsterdam, Acad Med Ctr, NL-1105 AZ Amsterdam, Netherlands
来源：
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2013年 / 56卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
P250
引用
收藏
页码：S337 / S337
页数：1
相关论文
共 50 条
  • [31] Quantification and Whole-Body Distribution of a Novel Dopamine D2/D3 Receptor Agonist, [18F]MCL-524, in Monkeys: A Prediction for Application in Human Subjects
    Finnema, S. J.
    Stepanov, V.
    Nakao, R.
    Amini, N.
    Sromek, A. W.
    Neumeyer, J. L.
    Seeman, P.
    Stabin, M. G.
    Farde, L.
    Halldin, C.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2012, 39 : S181 - S182
  • [32] In vitro characterisation of the high affinity D2/D3 dopamine agonist (+)PhNO
    Parker, Christine
    Clarke, K.
    Gee, A. D.
    Gee, A.
    Rabiner, E.
    NEUROIMAGE, 2006, 31 : T29 - T29
  • [33] Identification of novel dopamine D2 receptor ligands - a combined in silico / in vitro approach
    Zell, L.
    Kollar, J.
    Lainer, C.
    Temml, V.
    Schuster, D.
    FEBS OPEN BIO, 2022, 12 : 134 - 134
  • [34] Radiosynthesis of O-3-(2-[18F]fluoroethyl-L-DOPA ([18F]OFED) - a new fluorine-18 labeled phenylalanine derivative
    Kniess, Torsten
    Schroeder, Susann
    Hoepping, Alexander
    Zessin, Joerg
    Fuechtner, Frank
    Bergmann, Ralf
    Steinbach, Joerg
    JOURNAL OF NUCLEAR MEDICINE, 2016, 57
  • [35] Probing the D3R system using D2R knockout mice imaging with selective D3 agonist [18F] FHXPAT and D2/D3 antagonist [18F] fallypride
    Constantinescu, Cristian
    Mirbolooki, M. Reza
    Vikram, Bhatt
    Pan, Min-Liang
    Borrelli, Emiliana
    Mukherjee, Jogeshwar
    JOURNAL OF NUCLEAR MEDICINE, 2012, 53
  • [36] Radiosynthesis of F-18 labeled cytidine analog 2′-fluoro-5-iodo-l-β-D-arabinofuranosylcytosine ([18F]FIAC)
    Wu, Chun-Yi
    Chan, Pei-Chia
    Chang, Wei-Ting
    Liu, Ren-Shyan
    Alauddin, Mian M.
    Wang, Hsin-Ell
    APPLIED RADIATION AND ISOTOPES, 2009, 67 (7-8) : 1362 - 1365
  • [37] Synthesis and evaluation of 4-[18F] fluoropropoxy-3-iodobenzylguanidine ([18F]FPOIBG): A novel 18F-labeled analogue of MIBG
    Vaidyanathan, Ganesan
    McDougald, Darryl
    Koumarianou, Eftychia
    Choi, Jaeyeon
    Hens, Marc
    Zalutsky, Michael R.
    NUCLEAR MEDICINE AND BIOLOGY, 2015, 42 (08) : 673 - 684
  • [38] Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents
    Hocke, C
    Prante, O
    Löber, S
    Hübner, H
    Gmeiner, P
    Kuwert, T
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (21) : 4819 - 4823
  • [39] A Modified Simplified Reference Tissue Model for the Quantification of Dopamine D2/3 Receptors with [18F]Fallypride Images
    Tsartsalis, Stergios
    Moulin-Sallanon, Marcelle
    Dumas, Noe
    Tournier, Benjamin B.
    Ginovart, Nathalie
    Millet, Philippe
    MOLECULAR IMAGING, 2014, 13
  • [40] Synthesis, radiosynthesis and first in vitro evaluation of novel PET-tracers for the dopamine transporter: [11C]IPCIT and [18F]FE@IPCIT
    Rami-Mark, Christina
    Bornatowicz, Birgit
    Fink, Cornel
    Otter, Paul
    Ungersboeck, Johanna
    Vraka, Chrysoula
    Haeusler, Daniela
    Nics, Lukas
    Spreitzer, Helmut
    Hacker, Marcus
    Mitterhauser, Markus
    Wadsak, Wolfgang
    BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 21 (24) : 7562 - 7569
12345