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- [32] EFFICACY OF THE ORAL TYROSINE KINASE 2 (TYK2) INHIBITOR TAK-279 IN TWO PRECLINICAL MOUSE MODELS OF COLITISGASTROENTEROLOGY, 2024, 166 (05) : S1399 - S1399Kong, Kok-Fai论文数: 0 引用数: 0 h-index: 0Khan, Md A. Wadud论文数: 0 引用数: 0 h-index: 0Singh, Namita论文数: 0 引用数: 0 h-index: 0Van Anh Nguyen论文数: 0 引用数: 0 h-index: 0Wilson, Elizabeth论文数: 0 引用数: 0 h-index: 0Tang, Jay论文数: 0 引用数: 0 h-index: 0Marusic, Suzana论文数: 0 引用数: 0 h-index: 0Xia, Guliang论文数: 0 引用数: 0 h-index: 0Petrakis, Ioannis论文数: 0 引用数: 0 h-index: 0Nguyen, Deborah G.论文数: 0 引用数: 0 h-index: 0
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- [35] Highly Selective Inhibition of Tyrosine Kinase 2 (TYK2) for the Treatment of Autoimmune Diseases: Discovery of the Allosteric Inhibitor BMS-986165JOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (20) : 8973 - 8995Wrobleski, Stephen T.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAMoslin, Ryan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USALin, Shuqun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAZhang, Yanlei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USASpergel, Steven论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAKempson, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Dept Discovery Synth, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USATokarski, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAStrnad, Joann论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAZupa-Fernandez, Adriana论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USACheng, Lihong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAShuster, David论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAGillooly, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAYang, Xiaoxia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAHeimrich, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAMcIntyre, Kim W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAChaudhry, Charu论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Leads Discovery & Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAKhan, Javed论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USARuzanov, Max论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USATredup, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAMulligan, Dawn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAXie, Dianlin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Mol Struct & Design, Mol Discovery Technol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USASun, Huadong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAHuang, Christine论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAD'Arienzo, Celia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAAranibar, Nelly论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAChiney, Manoj论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAChimalakonda, Anjaneya论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Metab & Pharmacokinet Dept, Pharmaceut Candidate Optimizat, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAPitts, William J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USALombardo, Louis论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USABurke, James R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Biol, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USAWeinstein, David S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA Vividion Therapeut Inc, 5820 Nancy Ridge Dr, San Diego, CA 92121 USA Bristol Myers Squibb Res & Dev, Immunosci Discovery Chem, POB 4000, Princeton, NJ 08543 USA
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- [38] BMS-986165, an oral selective tyrosine kinase 2 (TYK2) inhibitor, does not affect the pharmacokinetics of methotrexate in healthy subjectsJOURNAL OF CROHNS & COLITIS, 2019, 13 : S437 - S438Chimalakonda, A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Princeton, NJ USAJones, J., III论文数: 0 引用数: 0 h-index: 0机构: PRA Hlth Sci, Blue Bell, PA USA Bristol Myers Squibb, Princeton, NJ USADockens, R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Princeton, NJ USAThroup, J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Princeton, NJ USABanerjee, S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Princeton, NJ USAGirgis, I.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Princeton, NJ USA Bristol Myers Squibb, Princeton, NJ USA
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- [40] BASELINE BIOMARKERS PREDICT BETTER RESPONSES TO DEUCRAVACITINIB, AN ORAL, SELECTIVE TYROSINE KINASE 2 (TYK2) INHIBITOR, IN A PHASE 2 TRIAL IN PSORIATIC ARTHRITISANNALS OF THE RHEUMATIC DISEASES, 2022, 81 : 215 - 216Fitzgerald, O.论文数: 0 引用数: 0 h-index: 0机构: Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, Ireland Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandGladman, D. D.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Rheumatol, Toronto, ON, Canada Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandMease, P. J.论文数: 0 引用数: 0 h-index: 0机构: Providence St Joseph Hlth, Swedish Med Ctr, Seattle, WA USA Univ Washington, Rheumatol Res, Seattle, WA 98195 USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandRitchlin, C. T.论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Allergy Immunol & Rheumatol, Rochester, NY 14627 USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandSmolen, J. S.论文数: 0 引用数: 0 h-index: 0机构: Med Univ Vienna, Rheumatol, Vienna, Austria Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandGao, L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Immunosci & Small Mol, Princeton, NJ USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandHu, S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Bioinformat, Princeton, NJ USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandNowak, M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Clin R&D, Princeton, NJ USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandBanerjee, S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rheumatol & Dermatol, Princeton, NJ USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, IrelandCatlett, I.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dermatol, Princeton, NJ USA Univ Coll Dublin UCD, Conway Inst, Rheumatol, Dublin, Ireland