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- [21] The Discovery, Preclinical, and Early Clinical Development of Potent and Selective GPR40 Agonists for the Treatment of Type 2 Diabetes Mellitus (LY2881835, LY2922083, and LY2922470)JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (24) : 10891 - 10916Hamdouchi, Chafiq论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAKahl, Steven D.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USALewis, Anjana Patel论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USACardona, Guemalli R.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAZink, Richard W.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAChen, Keyue论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAEessalu, Thomas E.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAFicorilli, James V.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAMarcelo, Marialuisa C.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAOtto, Keith A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAWilbur, Kelly L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USALineswala, Jayana P.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAPiper, Jared L.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USACoffey, D. Scott论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USASweetana, Stephanie A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAHaas, Joseph V.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USABrooks, Dawn A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAPratt, Edward J.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Singapore 237994, Singapore Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USABelin, Ruth M.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USADeeg, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAMa, Xiaosu论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USACannady, Ellen A.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAJohnson, Jason T.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAYumibe, Nathan P.论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAChen, Qi论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAMaiti, Pranab论文数: 0 引用数: 0 h-index: 0机构: Jubilant Biosys Res Ctr, Bangalore 560022, Karnataka, India Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAMontrose-Rafizadeh, Chahrzad论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAChen, Yanyun论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USAMiller, Anne Reifel论文数: 0 引用数: 0 h-index: 0机构: Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA Eli Lilly & Co, Lilly Corp Ctr, Div A, Lilly Res Labs, DC 0540, Indianapolis, IN 46285 USA
- [22] Discovery and Early Clinical Development of 2-{6-[2-(3,5-Dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a Soft-Drug Inhibitor of Phosphodiesterase 4 for Topical Treatment of Atopic DermatitisJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (14) : 5893 - 5903Felding, Jakob论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkSorensen, Morten D.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkPoulsen, Tina D.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkLarsen, Jens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkAndersson, Christina论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkRefer, Pia论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkEngell, Karen论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkLadefoged, Lotte G.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkThormann, Thorsten论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkVinggaard, Anne Marie论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkHegardt, Pontus论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkSohoel, Anders论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, DenmarkNielsen, Simon Feldbaek论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark LEO Pharma AS, New Prod Discovery & Global Dev, DK-2750 Ballerup, Denmark
- [23] Discovery and Early Clinical Development of Isobutyl 1-[8-Methoxy-5-(1-oxo-3H-isobenzofuran-5-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxylate (LEO 39652), a Novel "Dual-Soft" PDE4 Inhibitor for Topical Treatment of Atopic DermatitisJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (23) : 14502 - 14521Larsen, Jens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkLambert, Maja论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkPettersson, Henrik论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkVifian, Thomas论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkLarsen, Mogens论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkOllerstam, Anna论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkHegardt, Pontus论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Global Clin Operat Projects, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkEskilsson, Cecilia论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Preclin Dev, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkLaursen, Steen论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Preclin Dev, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkSoehoel, Anders论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Clin Pharmacol, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkSkak-Nielsen, Tine论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkHansen, Lene M.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Early Formulat & Analyt, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkKnudsen, Nina O.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Early Formulat & Analyt, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkEirefelt, Stefan论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkSorensen, Morten D.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkStilou, Tatiana G.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Skin Res, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, DenmarkNielsen, Simon F.论文数: 0 引用数: 0 h-index: 0机构: LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark LEO Pharma Global Res & Dev, Drug Design, DK-2750 Ballerup, Denmark