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- [11] Novel selective inhibitors of neutral endopeptidase: discovery by screening and hit-to-lead optimisationMEDCHEMCOMM, 2012, 3 (04) : 469 - 474El Bakali, Jamal论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceMaingot, Lucie论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceDumont, Julie论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceHost, Helene论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceHocine, Akila论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceCousaert, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceDassonneville, Sandrine论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceLeroux, Florence论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceDeprez, Benoit论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, FranceDeprez-Poulain, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France PRIM Pole Rech Interdisciplinaire Med, F-59006 Lille, France Univ Lille Nord France, Sch Pharm, INSERM, U761, F-59006 Lille, France
- [12] Discovery of pyrazolo[1,5-a]pyrimidin-7-amine derivatives as mTOR kinase domain inhibitors: Hit to lead optimizationABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248Deng, Yongqi论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USASun, Binyuan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAShipps, Gerald论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAMatthew, Richards论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAMeng, Zhaoyang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAWindsor, Williama论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAZeng, Hongbo论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USALong, Brian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USAXiao, Li论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Discovery, Boston, MA 02115 USA Merck Res Labs, Drug Discovery, Boston, MA 02115 USA
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- [14] HTS identification and optimization of Rho Kinase inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Hobson, Adrian D.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Worcester, MA USA Abbott Labs, Worcester, MA USA
- [15] Advantages of fluorinated fragment library in the discovery of novel specific binders and hit to lead optimizationABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2019, 258Gavrylenko, Oleksii论文数: 0 引用数: 0 h-index: 0机构: Chemspace, Monmouth Jct, NJ USA Chemspace, Monmouth Jct, NJ USAMoroz, Yurii论文数: 0 引用数: 0 h-index: 0机构: Chemspace, Monmouth Jct, NJ USA Chemspace, Monmouth Jct, NJ USA
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