Copper-catalyzed three-component one-pot synthesis of quinazolines

被引：53
|
作者：
Ju, Jia [1 ]
Hua, Ruimao [1 ,2 ]
Su, Ji [1 ]
机构：
[1] Tsinghua Univ, Dept Chem, Key Lab Organ Optoelect & Mol Engn, Minist Educ, Beijing 100084, Peoples R China
[2] Nankai Univ, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China
来源：
TETRAHEDRON | 2012年 / 68卷 / 46期
基金：
中国国家自然科学基金;
关键词：
Ammonia water; ortho-Bromo aromatic ketones; ortho-Bromo aromatic aldehydes; Aromatic aldehydes; Primary alcohols; Quinazolines; O-PHENYL OXIMES; 2-SUBSTITUTED QUINAZOLINES; DERIVATIVES; 2-PHENYLQUINAZOLINES; INHIBITORS;
D O I：
10.1016/j.tet.2012.09.035
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Two efficient approaches to multi-substituted quinazolines by the three-component one-pot reaction of o-bromo aromatic ketones/aldehydes, ammonia water and aromatic aldehydes, or primary alcohols catalyzed by CuCl have been developed. (C) 2012 Elsevier Ltd. All rights reserved.
引用
收藏
页码：9364 / 9370
页数：7
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