An improved synthesis of pyrazolines from aryl azides and acrylic esters

被引：0
|
作者：
Yadav, JS [1 ]
Reddy, BVS [1 ]
Geetha, V [1 ]
机构：
[1] Indian Inst Chem Technol, Hyderabad 500007, Andhra Pradesh, India
来源：
SYNLETT | 2002年 / 03期
关键词：
azides; Baylis-Hillman reaction; cycloaddition reactions; pyrazolines;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Substituted pyrazoline derivatives are synthesized in high yields through the cycloaddition reactions of azides with acrylates under Baylis-Hillman reaction conditions. Improved yields and enhanced rates are obtained using DABCO as the base.
引用
收藏
页码：513 / 515
页数：3
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