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- [21] The identification and pharmacological evaluation of potent, selective and orally available ACC1 inhibitorBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (23)Mizojiri, Ryo论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanAsano, Moriteru论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Otsuka Pharmaceut Factory Inc, Naruto, Tokushima 7728601, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanSasaki, Masako论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanSatoh, Yoshihiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Chordia Therapeut, Fujisawa, Kanagawa 2518585, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanYamamoto, Yukiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanSumi, Hiroyuki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Daiichi Sankyo Co LTD, Shinagawa Ku, Tokyo 1400005, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, JapanMaezaki, Hironobu论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan Axcelead Drug Discovery Partners Inc, Fujisawa, Kanagawa 2518585, Japan Takeda Pharmaceut Co Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2518555, Japan
- [22] Pharmacological characterization of the potent, selective and orally active cathepsin K inhibitor MIV-711BONE, 2012, 50 : S164 - S165Grabowska, U.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Saffron Walden, England Medivir, Saffron Walden, EnglandHenderson, I.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandEdlund, M.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandVrang, L.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandSedig, S.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandTerelius, Y.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandWikstrom, K.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandSahlberg, B. -L.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, EnglandChambers, T.论文数: 0 引用数: 0 h-index: 0机构: Univ London St Georges Hosp, London, England Medivir, Saffron Walden, EnglandLindstrom, E.论文数: 0 引用数: 0 h-index: 0机构: Medivir, Huddinge, Sweden Medivir, Saffron Walden, England
- [23] Discovery and preclinical evaluation of AMG 397, a potent, selective and orally bioavailable MCL1 inhibitorCANCER RESEARCH, 2020, 80 (16)Caenepeel, Sean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKaren, Rex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USABelmontes, Brian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAVerlinsky, Alla论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USATan, Hong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAChen, Xiaoyue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USALi, Kexue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAAllen, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAWahlstrom, Jan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USACoxon, Angela论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAHughes, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USA
- [24] The Novel TORC1/2 Kinase Inhibitor PQR620 Has Anti-Tumor Activity in Lymphomas as a Single Agent and in Combination with VenetoclaxCANCERS, 2019, 11 (06):Tarantelli, Chiara论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandGaudio, Eugenio论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandHillmann, Petra论文数: 0 引用数: 0 h-index: 0机构: PIQUR Therapeut AG, CH-4057 Basel, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandSpriano, Filippo论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandSartori, Giulio论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandAresu, Luca论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dipartimento Sci Vet, I-10095 Grugliasco, TO, Italy Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandCascione, Luciano论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland SIB, CH-1015 Lausanne, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland论文数: 引用数: h-index:机构:Kwee, Ivo论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland SIB, CH-1015 Lausanne, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandBeaufils, Florent论文数: 0 引用数: 0 h-index: 0机构: PIQUR Therapeut AG, CH-4057 Basel, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandZucca, Emanuele论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst Southern Switzerland, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandStathis, Anastasios论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst Southern Switzerland, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandWymann, Matthias P.论文数: 0 引用数: 0 h-index: 0机构: Univ Basel, Dept Biomed, CH-4056 Basel, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandCmiljanovic, Vladimir论文数: 0 引用数: 0 h-index: 0机构: PIQUR Therapeut AG, CH-4057 Basel, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandFabbro, Doriano论文数: 0 引用数: 0 h-index: 0机构: PIQUR Therapeut AG, CH-4057 Basel, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, SwitzerlandBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland Univ Svizzera Italiana, Inst Oncol Res, CH-6500 Bellinzona, Switzerland
- [25] Strategic Fluorination to Achieve a Potent, Selective, Metabolically Stable, and Orally Bioavailable Inhibitor of CSNK2MOLECULES, 2024, 29 (17):Ong, Han Wee论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAYang, Xuan论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USASmith, Jeffery L.论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USATaft-Benz, Sharon论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Genet, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAHowell, Stefanie论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USADickmander, Rebekah J.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Microbiol & Immunol, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAHavener, Tammy M.论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USASanders, Marcia K.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Genet, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USABrown, Jason W.论文数: 0 引用数: 0 h-index: 0机构: Takeda Dev Ctr Amer Inc, San Diego, CA 92121 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USACounago, Rafael M.论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, BR-13083875 Campinas, SP, Brazil Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAChang, Edcon论文数: 0 引用数: 0 h-index: 0机构: Takeda Dev Ctr Amer Inc, San Diego, CA 92121 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAKraemer, Andreas论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Inst Pharmaceut Chem, Struct Genom Consortium SGC, Max von Laue Str 9, D-60438 Frankfurt, Germany Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAMoorman, Nathaniel J.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Microbiol & Immunol, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA论文数: 引用数: h-index:机构:Axtman, Alison D.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USADrewry, David H.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USAWillson, Timothy M.论文数: 0 引用数: 0 h-index: 0机构: Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Struct Genom Consortium SGC, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Eshelman Sch Pharm, Div Chem Biol & Med Chem, Chapel Hill, NC 27599 USA Rapidly Emerging Antiviral Drug Dev Initiat READDI, Chapel Hill, NC 27599 USA
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