PHYSIOLOGICALLY BASED PHARMACOKINETIC (PBPK) MODELING OF ELAGOLIX FOR PREDICTION OF DRUG-DRUG INTERACTIONS (DDIS)

被引:0
|
作者
Chiney, M. S. [1 ]
Polepally, A. R. [1 ]
Nader, A. M. [1 ]
Dufek, M. B. [1 ]
Klein, C. E. [1 ]
Ng, J. W. [1 ]
Shebley, M. [1 ]
机构
[1] Abbvie, N Chicago, IL USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
PII-022
引用
收藏
页码:S59 / S59
页数:1
相关论文
共 50 条
  • [31] Prediction of pharmacokinetics and drug-drug interaction potential using physiologically based pharmacokinetic (PBPK) modeling approach: A case study of caffeine and ciprofloxacin
    Park, Min-Ho
    Shin, Seok-Ho
    Byeon, Jin-Ju
    Lee, Gwan-Ho
    Yu, Byung-Yong
    Shin, Young G.
    [J]. KOREAN JOURNAL OF PHYSIOLOGY & PHARMACOLOGY, 2017, 21 (01): : 107 - 115
  • [32] APPLICATION OF PHYSIOLOGICALLY BASED PHARMACOKINETIC (PBPK) MODELING FOR PREDICTION OF THE DRUG-DRUG INTERACTION (DDI) BETWEEN PAROXETINE AND TERBINAFINE IN A JAPANESE POPULATION.
    Yeo, K. Rowland
    Barter, Z.
    Almond, L.
    Rostami-Hodjegan, A.
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 2013, 93 : S119 - S120
  • [33] INVESTIGATING TRANSPORTER-MEDIATED DRUG-DRUG INTERACTIONS (DDIS) OF DASATINIB USING A PHYSIOLOGICALLY-BASED PHARMACOKINETIC MODEL.
    Chang, M.
    Bathena, S.
    Christopher, L.
    Shen, H.
    Roy, A.
    Leil, T.
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 2021, 109 : S7 - S7
  • [34] APPLICATION OF PHYSIOLOGICALLY BASED PHARMACOKINETIC (PBPK) MODELING FOR PREDICTION OF COMPLEX DRUG-DRUG INTERACTIONS (DDIs) INVOLVING OATPIB1-MEDIATED UPTAKE AND CYTOCHROME P450 (CYP) METABOLISM AND MULTIPLE INHIBITORS.
    Yeo, K. Rowland
    Jamei, M.
    Aarabi, M.
    Rostami-Hodjegan, A.
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 2012, 91 : S47 - S48
  • [35] Physiologically-based Pharmacokinetic (PBPK) Modelling of Transporter Medi-ated Drug Absorption, Clearance and Drug-drug Interactions
    Taskar, Kunal S.
    Harada, Isobel
    Alluri, Ravindra, V
    [J]. CURRENT DRUG METABOLISM, 2021, 22 (07) : 523 - 531
  • [36] Application of Physiologically Based Pharmacokinetic Modeling to Evaluate the Drug-Drug and Drug-Disease Interactions of Apatinib
    Liu, Hongrui
    Yu, Yiqun
    Guo, Nan
    Wang, Xiaojuan
    Han, Bing
    Xiang, Xiaoqiang
    [J]. FRONTIERS IN PHARMACOLOGY, 2021, 12
  • [37] APPLICATION OF PHYSIOLOGICALLY BASED PHARMACOKINETIC MODELING FOR PREDICTION OF CYP-MEDIATED DRUG-DRUG INTERACTIONS INVOLVING ETHINYLESTRADIOL.
    Ezuruike, U.
    Humphries, H.
    Dickins, M.
    Neuhoff, S.
    Gardner, I.
    Rowland-Yeo, K.
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 2018, 103 : S66 - S66
  • [38] Physiologically-Based Pharmacokinetic Modeling to Support the Clinical Management of Drug-Drug Interactions With Bictegravir
    Stader, Felix
    Battegay, Manuel
    Marzolini, Catia
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 2021, 110 (05) : 1231 - 1239
  • [39] Application of physiologically based pharmacokinetic modeling in predicting drug-drug interactions for sarpogrelate hydrochloride in humans
    Min, Jee Sun
    Kim, Doyun
    Park, Jung Bae
    Heo, Hyunjin
    Bae, Soo Hyeon
    Seo, Jae Hong
    Oh, Euichaul
    Bae, Soo Kyung
    [J]. DRUG DESIGN DEVELOPMENT AND THERAPY, 2016, 10 : 2959 - 2972
  • [40] Physiologically Based Pharmacokinetic Modeling for Selumetinib to Evaluate Drug-Drug Interactions and Pediatric Dose Regimens
    Cohen-Rabbie, Sarit
    Zhou, Li
    Vishwanathan, Karthick
    Wild, Martin
    Xu, Sherrie
    Freshwater, Tomoko
    Jain, Lokesh
    Schalkwijk, Stein
    Tomkinson, Helen
    Zhou, Diansong
    [J]. JOURNAL OF CLINICAL PHARMACOLOGY, 2021, 61 (11): : 1493 - 1504