Significant rate accelerated synthesis of glycosyl azides and glycosyl 1,2,3-triazole conjugates

被引：27

作者：

Kumar, Rishi ^{[1
]}

Maulik, Prakas R. ^{[1
]}

Misra, Anup Kumar ^{[1
]}

机构：

[1] Cent Drug Res Inst, Med & Proc Chem Div, Lucknow 226001, Uttar Pradesh, India

来源：

GLYCOCONJUGATE JOURNAL | 2008年 / 25卷 / 07期

关键词：

glycosyl azides; glycosyl triazoles; glycosyl bromides; click chemistry; one-pot;

D O I：

10.1007/s10719-007-9093-5

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

An efficient and significantly rapid access of a series of glycosyl azides and glycosyl 1,2,3-triazole conjugates is reported using modified one-pot reaction conditions. In both cases yields were excellent and single diastereomers were obtained.

引用

页码：595 / 602

页数：8

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