Synthesis and preclinical evaluation of carbon-11 labelled P2X7 receptor antagonists as PET tracers of microglial activation

被引：0

作者：

Janssen, Bieneke ^{[1
]}

Wilkinson, Shane M. ^{[2
]}

Ory, Dieter ^{[3
]}

Vugts, Danielle J. ^{[1
]}

van den Hoek, Johan J. ^{[1
]}

Schuit, Robert C. ^{[1
]}

Beaino, Wissam ^{[1
]}

Kooijman, Esther J. M. ^{[1
]}

Chishty, Mansoor ^{[4
]}

van der Perren, Anke ^{[5
]}

Baekelandt, Veerle ^{[5
]}

Molenaar, Ger T. ^{[1
,6
]}

Funke, Uta ^{[1
,6
]}

Shevchenko, Rostislav V. ^{[4
]}

Lammertsma, Adriaan A. ^{[1
]}

Bormans, Guy ^{[3
]}

Kassiou, Michael ^{[2
]}

Windhorst, Albert D. ^{[1
]}

机构：

[1] Vrije Univ Amsterdam Med Ctr, Radiol & Nucl Med, Amsterdam, Netherlands

[2] Univ Sydney, Sch Chem, Sydney, NSW, Australia

[3] Katholieke Univ Leuven, Lab Radiopharm, Dept Pharmaceut & Pharmacol Sci, Leuven, Belgium

[4] Pharmidex Pharmaceut Serv Ltd, London, England

[5] Katholieke Univ Leuven, Neurobiol & Gene Therapy, Dept Neurosci, Leuven, Belgium

[6] BV Cyclotron VU, Amsterdam, Netherlands

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2017年 / 60卷

关键词：

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

O 034

引用

页码：S53 / S53

页数：1

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