Synthesis of some new 2,3-diaryl-1,3-thiazolidin-4-ones as antibacterial agents

被引：49
|
作者：
Sayyed, M
Mokle, S
Bokhare, M
Mankar, A
Surwase, S
Bhusare, S [1 ]
Vibhute, Y
机构：
[1] Ysehwant Mahavidyalaya, Dept Chem, Nanded 431602, MS, India
[2] Shri Shivaji Coll, Dept Chem, Parbhani 431401, MS, India
来源：
ARKIVOC | 2006年
关键词：
4-amino-antipyrine; 4-amino-1,2,4-triazole; 2,6-dichloroaniline; 3-iodo-; and; 3-bromobenzaldehyde; thiazolidin-4-ones;
D O I：
10.3998/ark.5550190.0007.221
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Some new 2,3-diaryl-1,3-thiazolidin-4-one derivatives having a 2,6-dichlorophenyl, antipyrine, or 1,2,4-triazole ring at N-3 and variously substituted 3-iodo- or 3-bromo-phenyl rings at C-2 have been synthesized and tested as antibacterial agents. The results of the in vitro tests showed that some of them have effective antibacterial activity.
引用
下载
收藏
页码：187 / 192
页数：6
相关论文
共 50 条
  • [41] Synthesis of 5-arylidene-2-aryl-3-(benzotriazoloacetamidyl)-1,3-thiazolidin-4-ones as analegesic and antimicrobial agents
    Asati, KC
    Srivastava, SK
    Srivastava, SD
    INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 2006, 45 (02): : 526 - 531
  • [42] Microwave assisted synthesis and antibacterial study of 3-naphthyl-2-[(un)substituted phenyl]-1,3-thiazolidin-4-ones
    Chen, Hua
    Bai, Jie
    Zhao, Lian
    Yuan, Xiang-Guo
    Li, Xiao-Liu
    Cao, Ke-Qiang
    CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2008, 28 (06) : 1092 - 1096
  • [43] Microwave-assisted synthesis of 1,3-thiazolidin-4-ones and 2-aryl-1,3-oxathiolan-5-ones
    Cunico, Wilson
    Vellasco Junior, Walcimar T.
    Moreth, Marcele
    Gomes, Claudia R. B.
    LETTERS IN ORGANIC CHEMISTRY, 2008, 5 (05) : 349 - 352
  • [44] Synthesis and Antimycobacterial Activity of 2-aryl-3-(arylmethyl)-1,3-thiazolidin-4-ones
    Gomes, Claudia R. B.
    Moreth, Marcele
    Facchinetti, Victor
    de Souza, Marcus V. N.
    Vellasco Junior, Walcimar T.
    da Silva Lourenco, Maria Cristina
    Cunico, Wilson
    LETTERS IN DRUG DESIGN & DISCOVERY, 2010, 7 (05) : 353 - 358
  • [45] Discovery and optimization of 2,3-diaryl-1,3-thiazolidin-4-one-based derivatives as potent and selective cytotoxic agents with anti-inflammatory activity
    Shawky, Ahmed M.
    Almalki, Faisal A.
    Abdalla, Ashraf N.
    Youssif, Bahaa G. M.
    Abdel-Fattah, Maha M.
    Hersi, Fatima
    El-Sherief, Hany A. M.
    Nashwa, A. Ibrahim
    Gouda, Ahmed M.
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 259
  • [46] An efficient one-pot synthesis of new 2-imino-1,3-thiazolidin-4-ones under ultrasonic conditions
    Mamaghani, Manouchehr
    Loghmanifar, Azam
    Taati, Mohammad Reza
    ULTRASONICS SONOCHEMISTRY, 2011, 18 (01) : 45 - 48
  • [47] Synthesis of 5-arylidene-2-aryl-3-(2-chlorophenothiazinoacetamidyl)-1,3-thiazolidin-4-ones as antifungal and anticonvulsant agents
    Srivastava, SK
    Srivastava, SL
    Srivastava, SD
    JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 2000, 77 (02) : 104 - 105
  • [48] PARTITION-COEFFICIENTS AND CHROMATOGRAPHIC PARAMETERS OF SOME SUBSTITUTED 1,3-THIAZOLIDIN-4-ONES
    WOOLSTON, CRJ
    LEE, JB
    SWINBOURNE, FJ
    INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1994, 33 (06): : 590 - 592
  • [49] Topomer-CoMFA-based predictive modelling on 2,3-diaryl-substituted-1,3-thiazolidin-4-ones as non-nucleoside reverse transcriptase inhibitors
    Surendra Kumar
    Meena Tiwari
    Medicinal Chemistry Research, 2015, 24 : 245 - 257
  • [50] Topomer-CoMFA-based predictive modelling on 2,3-diaryl-substituted-1,3-thiazolidin-4-ones as non-nucleoside reverse transcriptase inhibitors
    Kumar, Surendra
    Tiwari, Meena
    MEDICINAL CHEMISTRY RESEARCH, 2015, 24 (01) : 245 - 257
12345