SYNTHESIS OF SOME 1,2,3-TRIAZOLES DERIVATIVES

被引:0
|
作者
Bouasla, Souad [1 ]
Fatmi, Chames Eddyn [1 ]
Teguiche, Mabrouk [1 ]
机构
[1] Guelma Univ, LCA, Fac Math Informat & Mat Sci, Dept Mat Sci, Guelma 24000, Algeria
关键词
aryl azides; DMAD; 1,3-dipolar cycloaddition; microwave irradiation; 1,2,3-triazoles; 1,3-DIPOLAR CYCLOADDITION; CHEMISTRY; EFFICIENT; SCIENCE; AZIDES;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Dimethyl acetylenedicarboxylate (DMAD) undergoes efficient Huisgen 1,3-dipolar cycloaddition reaction with various X-substituted aryl azides (X = 2Cl, 3Cl, 2COOCH(3), 4COOCH(3)), applying two different conditions, under conventional stirring at room temperature or under microwave irradiation, to afford the corresponding 1,4,5-trisubstituted 1,2,3-triazole 6-9 in good to excellent yields, especially when the phenyl ring of the azide is substituted at the ortho position.
引用
收藏
页码:1037 / 1040
页数:4
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