[11C]SNAP-7941, the first tracer for the melanin concentrating hormone receptor 1: Biodistribution and small animal PET

被引:0
|
作者
Philippe, Cecile [1 ,2 ]
Kuntner, Claudia [3 ]
Wanek, Thomas [3 ]
Mairinger, Severin [3 ]
Schirmer, Eva [4 ]
Spreitzer, Helmut [4 ]
Viernstein, Helmut [2 ]
Wadsak, Wolfgang [1 ,5 ]
Mitterhauser, Markus [1 ,2 ]
机构
[1] Med Univ Vienna, Dept Nucl Med, Radiochem & Biomarker Dev Unit, Vienna, Austria
[2] Univ Vienna, Dept Pharmaceut Technol & Biopharmaceut, A-1010 Vienna, Austria
[3] Austrian Inst Technol GmbH, Hlth & Environm Dept, Seibersdorf, Austria
[4] Univ Vienna, Dept Drug & Nat Prod Synth, A-1010 Vienna, Austria
[5] Univ Vienna, Dept Inorgan Chem, A-1010 Vienna, Austria
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
P332
引用
收藏
页码:S419 / S419
页数:1
相关论文
共 50 条
  • [41] PET measurements of Bmax and Kd with the k-opioid receptor tracer [11C]GR103545
    Tomasi, Giampaolo
    Nabulsi, Nabeel
    Weinzimmer, David
    Zeng, Ming-Quiang
    Blumberg, Laura
    Brown-Proctor, Clive
    Ding, Yu-Shin
    Carson, Richard
    Huang, Y.
    JOURNAL OF NUCLEAR MEDICINE, 2009, 50
  • [42] Small animal PET imaging of myocardial PDE4 with (R)-[11C]rolipram in rats
    Thomas, Adam
    Renaud, Jennifer
    Lortie, Mireille
    Kenk, Miran
    Thorn, Stephanie
    Beanlands, Robert
    DaSilva, Jean
    deKemp, Robert
    JOURNAL OF NUCLEAR MEDICINE, 2010, 51
  • [43] Modeling analysis of the CB1 PET tracer [11C]OMAR in rhesus monkeys and humans
    Normandin, Marc D.
    Weinzimmer, David P.
    Ropchan, Jim
    Labaree, David
    Lin, Kuo-Shyan
    Mason, Neale S.
    Carson, Richard E.
    D'Souza, Deepak C.
    Neumeister, Alexander
    Huang, Yiyun
    NEUROIMAGE, 2010, 52 : S13 - S13
  • [44] Kinetic modeling of CB1 PET tracer [11C]OMAR in rhesus monkeys and humans
    Normandin, Marc
    Weinzimmer, David
    Ropchan, Jim
    Labaree, David
    Lin, Kuo-Shyan
    Mason, Neale
    Carson, Richard
    D'Souza, Deepak
    Neumeister, Alexander
    Huang, Yiyun
    JOURNAL OF NUCLEAR MEDICINE, 2010, 51
  • [45] Biodistribution and dosimetry of the GluN2B-specific NMDA receptor PET radioligand (R)-[11C]Me-NB1
    Rischka, Lucas
    Murgas, Matej
    Pichler, Verena
    Vraka, Chrysoula
    Rausch, Ivo
    Winkler, Dietmar
    Nics, Lukas
    Rasul, Sazan
    Silberbauer, Leo Robert
    Reed, Murray Bruce
    Godbersen, Godber Mathis
    Unterholzner, Jakob
    Handschuh, Patricia
    Gryglewski, Gregor
    Mindt, Thomas
    Mitterhauser, Markus
    Hahn, Andreas
    Ametamey, Simon Mensah
    Wadsak, Wolfgang
    Lanzenberger, Rupert
    Hacker, Marcus
    EJNMMI RESEARCH, 2022, 12 (01)
  • [46] Biodistribution and dosimetry of the GluN2B-specific NMDA receptor PET radioligand (R)-[11C]Me-NB1
    Lucas Rischka
    Matej Murgaš
    Verena Pichler
    Chrysoula Vraka
    Ivo Rausch
    Dietmar Winkler
    Lukas Nics
    Sazan Rasul
    Leo Robert Silberbauer
    Murray Bruce Reed
    Godber Mathis Godbersen
    Jakob Unterholzner
    Patricia Handschuh
    Gregor Gryglewski
    Thomas Mindt
    Markus Mitterhauser
    Andreas Hahn
    Simon Mensah Ametamey
    Wolfgang Wadsak
    Rupert Lanzenberger
    Marcus Hacker
    EJNMMI Research, 12
  • [47] Small molecule melanin-concentrating hormone receptor 1 (MCH1R) antagonists as anxiolytic and antidepressive agents
    Dyck, B
    DRUG DEVELOPMENT RESEARCH, 2005, 65 (04) : 291 - 300
  • [48] Synthesis and initial evaluation of [11C]JNJ7777120 as a PET tracer for the histamine H4 receptor
    Funke, Uta
    Smits, Rogier A.
    Mooijer, Martien P. J.
    Verlaan, Mariska
    Verbeek, Joost
    Vugts, Danielle J.
    Spaans, Arnold
    Janssen, Bieneke
    Lammertsma, Adriaan A.
    Kruijer, Perry S.
    Leurs, Rob
    Perk, Lars R.
    Windhorst, Albert D.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2013, 56 : S81 - S81
  • [49] Pre-clinical evaluations of novel peripheral benzodiazepine receptor PET tracer [11C]DAA1106
    Maeda, J
    Zhang, MR
    Okauchi, T
    Ikoma, Y
    Suzuki, K
    Suhara, T
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2004, 94 : 299P - 299P
  • [50] In vivo biodistribution, biokinetics and blood metabolism of 11C-PK11195 in rats - a PET tracer for peripheral benzodiazepine receptor
    Virsu, P.
    Laitinen, I.
    Poyhonen, T.
    Nagren, K.
    Roivainen, A.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2005, 32 : S266 - S266