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- [39] IRREVERSIBLE ENZYME INHIBITORS . 136 . 2,4- DIAMINO-5-(3,4-DICHLOROPHENYL)-6-(P-(M-FLUOROSULFONYLBENZAMIDO)PHENOXYMETHYL)PYRIMIDINE AN ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITOR OF DIHYDROFOLIC REDUCTASE . EFFECT OF STRUCTURE ON ISOZYME SPECIFICITY JOURNAL OF MEDICINAL CHEMISTRY, 1969, 12 (01) : 82 - +