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- [1] Novel pyrrolopyrimidines as Mps1/TTK kinase inhibitors for breast cancerBIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (07) : 2156 - 2166Sugimoto, Yasuro论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USASawant, Dwitiya B.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Arts & Sci, Dept Mol Genet, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAFisk, Harold A.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Arts & Sci, Dept Mol Genet, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAMao, Liguang论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USALi, Chenglong论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USAChettiar, Somsundaram论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA论文数: 引用数: h-index:机构:Darby, Michael V.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USABrueggemeier, Robert W.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA Ohio State Univ, Coll Pharm, Div Med Chem & Pharmacognosy, Columbus, OH 43210 USA
- [2] Development of the First Covalent Monopolar Spindle Kinase 1 (MPS1/TTK) InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (04) : 3173 - 3192Serafim, Ricardo A. M.论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanySantiago, Andre da Silva论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany论文数: 引用数: h-index:机构:Hu, Zexi论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Tubingen, Dept Med Oncol & Pneumol Internal Med 8, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & F, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germanydos Reis, Caio, V论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyTakarada, Jessica E.论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyMezzomo, Priscila论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyMassirer, Katlin B.论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyKudolo, Mark论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyGerstenecker, Stefan论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany论文数: 引用数: h-index:机构:Zender, Lars论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Tubingen, Dept Med Oncol & Pneumol Internal Med 8, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & F, D-72076 Tubingen, Germany German Canc Res Ctr, German Consortium Translat Canc Res DKTK, Partner Site Tubingen, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyKnapp, Stefan论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt, Buchmann Inst Mol Life Sci, Struct Genom Consortium, D-60438 Frankfurt, Germany Goethe Univ Frankfurt, Inst Pharmaceut Chem, Buchmann Inst Mol Life Sci, D-60438 Frankfurt, Germany Frankfurt Canc Inst FCI, Site Frankfurt Mainz, D-60596 Frankfurt, Germany German Translat Canc Network DKTK, Site Frankfurt Mainz, D-60596 Frankfurt, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyLaufer, Stefan论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & F, D-72076 Tubingen, Germany Tubingen Ctr Acad Drug Discovery, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyCounago, Rafael M.论文数: 0 引用数: 0 h-index: 0机构: Univ Estadual Campinas, Ctr Biol Mol & Engn Genet CBMEG, Ctr Quim Med CQMED, UNICAMP, BR-13083875 Campinas, SP, Brazil Univ Estadual Campinas, Inst Biol, Dept Genet & Evolucao, Struct Genom Consortium, BR-13083886 Campinas, SP, Brazil Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, GermanyGehringer, Matthias论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany Univ Tubingen, Cluster Excellence iFIT EXC 2180 Image Guided & F, D-72076 Tubingen, Germany Eberhard Karls Univ Tubingen, Dept Pharmaceut Med Chem, D-72076 Tubingen, Germany
- [3] Mps1/TTK: a novel target and biomarker for cancerJOURNAL OF DRUG TARGETING, 2017, 25 (02) : 112 - 118Xie, Yuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaWang, Anqiang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaLin, Jianzhen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaWu, Liangcai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaZhang, Haohai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaYang, Xiaobo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaWan, Xueshuai论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaMiao, Ruoyu论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Beth Israel Deaconess Med Ctr, Liver Ctr & Transplant Inst, Dept Med, Boston, MA USA Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaSang, Xinting论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R ChinaZhao, Haitao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China Peking Union Med Coll, 1 Shuaifuyuan, Beijing 100730, Peoples R China Chinese Acad Med Sci, Peking Union Med Coll Hosp, Dept Liver Surg, 1 Shuaifuyuan, Beijing 100730, Peoples R China
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- [9] Inhibition of mitotic kinase Mps1 promotes cell death in neuroblastomaScientific Reports, 10Sonia Simon Serrano论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of MedicineWondossen Sime论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of MedicineYasmin Abassi论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of MedicineRenée Daams论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of MedicineRamin Massoumi论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of MedicineMohamed Jemaà论文数: 0 引用数: 0 h-index: 0机构: Lund University,Department of Laboratory Medicine, Translational Cancer Research, Faculty of Medicine
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