Efficient synthesis of C-11 functionalized steroids

被引：6
|
作者：
Bazzini, Patrick
Ibrahim-Ouali, Malika
Pellissier, Helene
Santelli, Maurice
机构：
[1] CNRS, UMR 6180, F-13397 Marseille 20, France
[2] Univ Aix Marseille 3, CNRS, Fac Sci & Tech St Jerome, Lab Synthese Organ Associe, Marseille 20, France
来源：
STEROIDS | 2006年 / 71卷 / 06期
关键词：
non-natural steroids; functionalization; C-11 substituted steroids;
D O I：
10.1016/j.steroids.2006.01.003
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
An efficient synthesis from readily available materials of numerous steroids functionalized at C-11 position, interesting from a biological point of view, is described using our general approach. The characteristic H-1 and C-13 NMR spectroscopic features of the synthesized steroids are reported. (c) 2006 Elsevier Inc. All rights reserved.
引用
收藏
页码：459 / 468
页数：10
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