Quinazoline and quinoline derivatives as inhibitors of adaptor associated kinase 1

被引:0
|
作者
Hartz, Richard [1 ]
Ahuja, Vijay [2 ]
Dzierba, Carolyn [1 ]
Dasgupta, Bireshwar [1 ]
Kostich, Walter [1 ]
Nara, Susheel [3 ]
Easton, Amy [1 ]
Bourin, Clotilde [1 ]
Bristow, Linda [1 ]
Brown, Jeffrey [1 ]
Hunihan, Lisa [1 ]
Gulianello, Michael [1 ]
Westphal, Ryan [1 ]
Rajamani, Ramkumar [1 ]
Kiefer, Susan [2 ]
Camac, Dan [2 ]
Muckelbauer, Jodi [2 ]
Pokross, Matt [2 ]
Mannan, Vijayakumar Chittor [3 ]
Manepalli, Raju [3 ]
Sarvasiddhi, Sarat [3 ]
Honkhambe, Swarnamba [3 ]
Kandula, Sathaiah [3 ]
Patankar, Vidya [3 ]
Brown, Randi [1 ]
Surti, Neha [1 ]
Lippy, Jonathan [2 ]
Padmanabha, Ramesh [1 ]
Esposito, Kim [1 ]
Hamman, Brian [4 ]
Allen, Jason [4 ]
Baker, Kevin [4 ]
Savelieva, Katerina [4 ]
Zambrowicz, Brian [4 ]
Pattipati, Sreenivasulu [3 ]
Dokania, Manoj [3 ]
Elavazhagan, Saravanan [3 ]
Dandapani, Kumaran [3 ]
Bronson, Joanne [1 ]
Macor, John [2 ]
机构
[1] Bristol Myers Squibb, Wallingford, CT USA
[2] Bristol Myers Squibb, Princeton, NJ USA
[3] Syngene Int, Bangalore, Karnataka, India
[4] Lexicon Pharmaceut, Princeton, NJ USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
395
引用
下载
收藏
页数:1
相关论文
共 50 条
  • [1] Molecular design and synthesis of inhibitors of EGFR kinase: New quinazoline derivatives
    Bunev, Alexander
    Sukhonosova, Elena
    Sokov, Sergey
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253
  • [2] A patent review of adaptor associated kinase 1 (AAK1) inhibitors (2013-present)
    Martinez-Gualda, Belen
    Schols, Dominique
    De Jonghe, Steven
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2021, 31 (10) : 911 - 936
  • [3] Research progress in quinazoline derivatives as multi-target tyrosine kinase inhibitors
    Jin, Hao
    Dan, Hu-Guang
    Rao, Guo-Wu
    HETEROCYCLIC COMMUNICATIONS, 2018, 24 (01) : 1 - 10
  • [4] Synthesis, Characterization, and DFT Calculations of Quinoline and Quinazoline Derivatives
    H. S. Mohamed
    M. K. Abdel-Latif
    S.A. Ahmed
    Russian Journal of Organic Chemistry, 2020, 56 : 1660 - 1668
  • [5] Synthesis, Characterization, and DFT Calculations of Quinoline and Quinazoline Derivatives
    Mohamed, H. S.
    Abdel-Latif, M. K.
    Ahmed, S. A.
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2020, 56 (09) : 1660 - 1668
  • [6] Development and therapeutic potential of adaptor-associated kinase 1 inhibitors in human multifaceted diseases
    Xin, Xin
    Wang, Yue
    Zhang, Lele
    Zhang, Dan
    Sha, Leihao
    Zhu, Ziyu
    Huang, Xiaoyi
    Mao, Wuyu
    Zhang, Jifa
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 248
  • [7] Quinazoline derivatives as selective CYP1B1 inhibitors
    Siddique, Mohd Usman Mohd
    McCann, Glen J. P.
    Sonawane, Vinay R.
    Horley, Neill
    Gatchie, Linda
    Joshi, Prashant
    Bharate, Sandip B.
    Jayaprakash, Venkatesan
    Sinha, Barij N.
    Chaudhuri, Bhabatosh
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 130 : 320 - 327
  • [8] Discovery of novel quinazoline derivatives bearing semicarbazone moiety as potent EGFR kinase inhibitors
    Tu, Yuanbiao
    Wang, Caolin
    Yang, Zunhua
    Zhao, Bingbing
    Lai, Luogen
    Yang, Qi
    Zheng, Pengwu
    Zhu, Wufu
    COMPUTATIONAL AND STRUCTURAL BIOTECHNOLOGY JOURNAL, 2018, 16 : 462 - 478
  • [9] Sulfonylated Indeno[1,2-c]quinoline Derivatives as Potent EGFR Tyrosine Kinase Inhibitors
    Hengphasatporn, Kowit
    Aiebchun, Thitinan
    Mahalapbutr, Panupong
    Auepattanapong, Atima
    Khaikate, Onnicha
    Choowongkomon, Kiattawee
    Kuhakarn, Chutima
    Meesin, Jatuporn
    Shigeta, Yasuteru
    Rungrotmongkol, Thanyada
    ACS OMEGA, 2023, 8 (22): : 19645 - 19655
  • [10] Synthesis and Characterization of Quinoline-3-Carboxamide Derivatives as Inhibitors of the ATM Kinase
    Ravi, Srimadhavi
    Barui, Sugata
    Kirubakaran, Sivapriya
    Duhan, Parul
    Bhowmik, Kaushik
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2020, 20 (23) : 2070 - 2079