Microwave promoted Suzuki cross-coupling reactions of quinazoline halides with aryl boronic acids

被引:0
|
作者
Akula, Kalyan Chakravarthy [1 ]
Chakka, Ramesh [1 ]
Puri, Usha Rani [1 ]
Kunamalla, Deepa Kranthi [1 ]
机构
[1] Dr Reddys Labs Ltd, Hyderabad 500016, Andhra Pradesh, India
关键词
microwave synthesis; Suzuki cross-coupling reactions; quinazoline halides; aryl boronic acids;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
The microwave promoted Suzuki coupling reaction of quinazoline halides with boronic acids performed was studied using stable catalyst tetrakis triphenyl phosphine palladium (0). This catalyst under microwave conditions (175 degrees C, 6 m) provided coupled products with yields ranging from 76 to 90 %. This method tolerated a variety of boronic acids in the absence of ligand.
引用
收藏
页码:119 / 124
页数:6
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