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- [1] Mutations in UBA3 Confer Resistance to the NEDD8-Activating Enzyme Inhibitor MLN4924 in Human Leukemic Cells[J]. PLOS ONE, 2014, 9 (04):Xu, G. Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaToth, Julia I.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, NCI Designated Canc Ctr, La Jolla, CA 92037 USA Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canadada Silva, Sara R.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Dept Chem, Mississauga, ON L5L 1C6, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaPaiva, Stacey-Lynn论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Dept Chem, Mississauga, ON L5L 1C6, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaLukkarila, Julie L.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Dept Chem, Mississauga, ON L5L 1C6, Canada Sheridan Inst Technol & Adv Learning, HalTech Reg Innovat Ctr, Oakville, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaHurren, Rose论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaMaclean, Neil论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaSukhai, Mahadeo A.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaBhattacharjee, Rabindra N.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaGoard, Carolyn A.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaGunning, Patrick T.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Dept Chem, Mississauga, ON L5L 1C6, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaDhe-Paganon, Sirano论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Childrens Hosp, Sch Med, Div Nephrol, Boston, MA 02115 USA Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaPetroski, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, NCI Designated Canc Ctr, La Jolla, CA 92037 USA Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, CanadaSchimmer, Aaron D.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada Univ Hlth Network, Princess Margaret Canc Ctr, Ontario Canc Inst, Toronto, ON, Canada
- [2] Mutations in UBA3 Confer Resistance to the NEDD8-Activating Enzyme Inhibitor MLN4924 in Human Leukemic Cells (vol 9, e93530, 2014)[J]. PLOS ONE, 2014, 9 (10):Xu, G. W.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USAToth, J., I论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USAda Silva, S. R.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USAPaiva, S-L论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USALukkarila, J. L.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA Stanford Univ, Sch Med, Div Hematol, Stanford, CA 94305 USA论文数: 引用数: h-index:机构:
- [3] Treatment-Emergent Mutations in NAEβ Confer Resistance to the NEDD8-Activating Enzyme Inhibitor MLN4924[J]. CANCER CELL, 2012, 21 (03) : 388 - 401Milhollen, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAThomas, Michael P.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USANarayanan, Usha论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USATraore, Tary论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USARiceberg, Jessica论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAAmidon, Benjamin S.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USABence, Neil F.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USABolen, Joseph B.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USABrownell, James论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USADick, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USALoke, Huay-Keng论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAMcDonald, Alice A.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAMa, Jingya论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAManfredi, Mark G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USASells, Todd B.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USASintchak, Mike D.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAYang, Xiaofeng论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAXu, Qing论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAKoenig, Erik M.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USAGavin, James M.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Discovery, Cambridge, MA 02139 USA
- [4] Radiosensitization of Human Colorectal Cancer Cells by MLN4924: An Inhibitor of NEDD8-Activating Enzyme[J]. TECHNOLOGY IN CANCER RESEARCH & TREATMENT, 2016, 15 (04) : 527 - 534论文数: 引用数: h-index:机构:Zhu, Ji论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R ChinaLi, Guichao论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R ChinaZhang, Zhen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China
- [5] Radiosensitization of Human Pancreatic Cancer Cells by MLN4924, an Investigational NEDD8-Activating Enzyme Inhibitor[J]. CANCER RESEARCH, 2012, 72 (01) : 282 - 293Wei, Dongping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALi, Hua论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAYu, Jie论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASebolt, Jonathan T.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAZhao, Lili论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALawrence, Theodore S.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAMorgan, Meredith A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASun, Yi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA
- [6] Mechanistic RBC Partitioning Studies of MLN4924, a Nedd8-Activating Enzyme inhibitor[J]. DRUG METABOLISM REVIEWS, 2010, 42 : 94 - 95Xia, Cindy Q.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USAChen, Susan论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USAZhang, Ji论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USAWu, Jing-Tao论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USAQian, Mark G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USALee, Frank W.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USABalani, Suresh K.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA Millennium Pharmaceut Inc, Dmpk, Cambridge, MA USA
- [7] A Gatekeeper Residue for NEDD8-Activating Enzyme Inhibition by MLN4924[J]. CELL REPORTS, 2012, 1 (04): : 309 - 316Toth, Julia I.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USAYang, Li论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USADahl, Russell论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USAPetroski, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA
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Lab Transplant Engn & Immunol, Sichuan Prov Engn Lab Pathol Clin Applicat, Chengdu 610041, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaGeng, Xue论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Cao, Yongliang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, 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Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaHu, Yue论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China论文数: 引用数: h-index:机构:Yin, Xuhui论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Inst Neurosci, Zhengzhou 450052, Peoples R China Zhengzhou Univ, Affiliated Hosp 3, Zhengzhou 450052, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaRan, Yunwei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Inst Neurosci, Zhengzhou 450052, Peoples R China Zhengzhou Univ, Affiliated Hosp 3, Zhengzhou 450052, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaYang, Hao论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, Inst Syst Genet, Chengdu 610041, Peoples R China Sichuan Univ, West China Hosp, NHC Key Lab Transplant Engn & Immunol, Sichuan Prov Engn Lab Pathol Clin Applicat, Chengdu 610041, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaFan, Wenying论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaZhao, Bing-Qiao论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, 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