共 50 条
- [1] A Gatekeeper Residue for NEDD8-Activating Enzyme Inhibition by MLN4924[J]. CELL REPORTS, 2012, 1 (04): : 309 - 316Toth, Julia I.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USAYang, Li论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USADahl, Russell论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USAPetroski, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA Sanford Burnham Med Res Inst, Signal Transduct Program, La Jolla, CA 92037 USA
- [2] The NEDD8-activating enzyme inhibitor MLN4924 reduces ischemic brain injury in mice[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 119 (06)Yu, Huilin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaLuo, Haiyu论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaChang, Luping论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaWang, Shisheng论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, Inst Syst Genet, Chengdu 610041, Peoples R China Sichuan Univ, West China Hosp, NHC Key Lab Transplant Engn & Immunol, Sichuan Prov Engn Lab Pathol Clin Applicat, Chengdu 610041, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaGeng, Xue论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaKang, Lijing论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaZhong, Yi论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, Inst Syst Genet, Chengdu 610041, Peoples R China Sichuan Univ, West China Hosp, NHC Key Lab Transplant Engn & Immunol, Sichuan Prov Engn Lab Pathol Clin Applicat, Chengdu 610041, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaCao, Yongliang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaWang, Ranran论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaYang, Xing论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaZhu, Yuanbo论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaShi, Mei-Juan论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaHu, Yue论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaLiu, Zhongwang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaYin, Xuhui论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Inst Neurosci, Zhengzhou 450052, Peoples R China Zhengzhou Univ, Affiliated Hosp 3, Zhengzhou 450052, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaRan, Yunwei论文数: 0 引用数: 0 h-index: 0机构: Zhengzhou Univ, Inst Neurosci, Zhengzhou 450052, Peoples R China Zhengzhou Univ, Affiliated Hosp 3, Zhengzhou 450052, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaYang, Hao论文数: 0 引用数: 0 h-index: 0机构: Sichuan Univ, Inst Syst Genet, Chengdu 610041, Peoples R China Sichuan Univ, West China Hosp, NHC Key Lab Transplant Engn & Immunol, Sichuan Prov Engn Lab Pathol Clin Applicat, Chengdu 610041, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaFan, Wenying论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R ChinaZhao, Bing-Qiao论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China Fudan Univ, Inst Brain Sci, MOE Frontiers Ctr Brain Sci, Shanghai 200032, Peoples R China Fudan Univ, Jingan Dist Ctr Hosp Shanghai, Inst Brain Sci, State Key Lab Med Neurobiol, Shanghai 200032, Peoples R China
- [3] Radiosensitization of Human Colorectal Cancer Cells by MLN4924: An Inhibitor of NEDD8-Activating Enzyme[J]. TECHNOLOGY IN CANCER RESEARCH & TREATMENT, 2016, 15 (04) : 527 - 534Wan, Juefeng论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R ChinaZhu, Ji论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R ChinaLi, Guichao论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R ChinaZhang, Zhen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China Fudan Univ, Shanghai Med Coll, Dept Oncol, Shanghai, Peoples R China Fudan Univ, Dept Radiat Oncol, Shanghai Canc Ctr, 270 Dong An Rd, Shanghai 200032, Peoples R China
- [4] Discovery of the Nedd8 activating enzyme inhibitor MLN4924[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Langston, Steven P.论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Int Co, Dept Oncol Chem, Cambridge, MA 02139 USA Takeda Pharmaceut Int Co, Dept Oncol Chem, Cambridge, MA 02139 USA
- [5] Targeting the protein ubiquitination machinery in melanoma by the NEDD8-activating enzyme inhibitor pevonedistat (MLN4924)[J]. INVESTIGATIONAL NEW DRUGS, 2017, 35 (01) : 11 - 25论文数: 引用数: h-index:机构:Micel, Lindsey N.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USASelby, Heather M.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USATan, Aik Choon论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Colorado, Ctr Canc, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USAPitts, Todd M.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Colorado, Ctr Canc, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USABagby, Stacey M.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USASpreafico, Anna论文数: 0 引用数: 0 h-index: 0机构: Princess Margaret Canc Ctr, Dept Med Oncol, Toronto, ON, Canada Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USAKlauck, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USABlakemore, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USASmith, Peter F.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USAMcDonald, Alice论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USABerger, Allison论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USATentler, John J.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Colorado, Ctr Canc, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USAEckhardt, S. Gail论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Dept Med, Div Med Oncol, Dev Therapeut Program, Anschutz Med Campus, Aurora, CO 80045 USA Univ Colorado, Ctr Canc, Aurora, CO 80045 USA Univ Washington, Sch Med, Dept Med, Div Med Oncol, Seattle, WA 98195 USA
- [6] The NEDD8-Activating Enzyme Inhibitor MLN4924 Disrupts Nucleotide Metabolism and Augments the Efficacy of Cytarabine[J]. CLINICAL CANCER RESEARCH, 2015, 21 (02) : 439 - 447Nawrocki, Steffan T.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USAKelly, Kevin R.论文数: 0 引用数: 0 h-index: 0机构: USC, Kenneth Norris Jr Comprehens Canc Ctr, Pasadena, CA USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA H3 Biomed, Cambridge, MA USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USAKeaton, Mignon论文数: 0 引用数: 0 h-index: 0机构: Metabolon Inc, Durham, NC USA Duke Univ, Durham, NC USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USACarraway, Hetty论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44195 USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USASekeres, Mikkael A.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44195 USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USAMaciejewski, Jaroslaw P.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44195 USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USACarew, Jennifer S.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Taussig Canc Inst, Cleveland, OH 44195 USA Univ Texas Hlth Sci Ctr San Antonio, CTRC, Div Hematol Oncol, San Antonio, TX 78229 USA
- [7] Targeting the protein ubiquitination machinery in melanoma by the NEDD8-activating enzyme inhibitor pevonedistat (MLN4924)[J]. Investigational New Drugs, 2017, 35 : 11 - 25Kit Man Wong论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineLindsey N. Micel论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineHeather M. Selby论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineAik Choon Tan论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineTodd M. Pitts论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineStacey M. Bagby论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineAnna Spreafico论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicinePeter J. Klauck论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineStephen J. Blakemore论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicinePeter F. Smith论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineAlice McDonald论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineAllison Berger论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineJohn J. Tentler论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of MedicineS. Gail Eckhardt论文数: 0 引用数: 0 h-index: 0机构: University of Washington School of Medicine,Division of Medical Oncology, Department of Medicine
- [8] MLN4924: a novel first-in-class inhibitor of NEDD8-activating enzyme for cancer therapy[J]. EXPERT OPINION ON INVESTIGATIONAL DRUGS, 2012, 21 (10) : 1563 - 1573Nawrocki, Steffan T.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USA Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USAGriffin, Patrick论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USA Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USAKelly, Kevin R.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USA Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USACarew, Jennifer S.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USA Univ Texas Hlth Sci Ctr San Antonio, Canc Therapy & Res Ctr, San Antonio, TX 78229 USA
- [9] Radiosensitization of Human Pancreatic Cancer Cells by MLN4924, an Investigational NEDD8-Activating Enzyme Inhibitor[J]. CANCER RESEARCH, 2012, 72 (01) : 282 - 293Wei, Dongping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALi, Hua论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAYu, Jie论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASebolt, Jonathan T.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAZhao, Lili论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USALawrence, Theodore S.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASmith, Peter G.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USAMorgan, Meredith A.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USASun, Yi论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Div Radiat & Canc Biol, Dept Radiat Oncol, Ann Arbor, MI 48109 USA
- [10] Quantifiable analysis of cellular pathway inhibition of a Nedd8-activating enzyme inhibitor, MLN4924, using AlphaScreen[J]. ANALYTICAL BIOCHEMISTRY, 2013, 439 (02) : 109 - 115Yan, Zhong-Hua论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABurkhardt, Anne论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USALoke, Huay-Keng论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAChen, Jesse论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAXu, Qing论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABrauer, Pam论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAMa, Jingya论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USALin, Yafang论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USAGarcia, Khris论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USADick, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USABembenek, Michael E.论文数: 0 引用数: 0 h-index: 0机构: Millennium Pharmaceut Inc, Cambridge, MA 02139 USA Millennium Pharmaceut Inc, Cambridge, MA 02139 USA