SYNTHESIS OF 3-[2-(SUBSTITUTED SULFONYL)-1H-IMIDAZOL-YL] CHROMEN-2-ONE DERIVATIVES

被引:0
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作者
Guravaiah, Nalajam [1 ]
Rao, Vedula Rajeswar [1 ]
机构
[1] Natl Inst Technol, Dept Chem, Warangal 506021, Andhra Pradesh, India
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Reaction of 3-(2-Mercapto-1H-imidazol-4-yl)chromen-2-one (1) with various alkyl/aryl/phenacyl halides in a mixture of anhydrous ethanol and dimethyl formamide gave the corresponding 3-(2-substituted sulfanyl-1H-imidazol-4-yl)chromen-2-ones (2). These on further reaction with hydrogen peroxide in acetic acid resulted in the formation of corresponding sulfones(3) in good yields the structure of the synthesized compounds were established from evidences like IR,NMR and mass spectral data.
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页码:367 / 374
页数:8
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