3-Aminopyrroles and their application in the synthesis of pyrrolo[3,2-d]pyrimidine (9-deazapurine) derivatives

被引：0
|
作者：
Salaheldin, Abdellatif M. [1 ]
Oliveira-Campos, Ana M. F. [1 ]
Rodrigues, Ligia M. [1 ]
机构：
[1] Univ Minho, IBQF, Ctr Quim, P-4710057 Braga, Portugal
来源：
ARKIVOC | 2008年
关键词：
3-Aminopyrrole; pyrrolo[3,2-d] pyrimidine; 9-deazapurines; beta-enaminonitriles; Thorpe-Ziegler cyclization;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
3-Aminopyrrole derivatives have been synthesized from 3-anilino-2-cyanoacrylonitrile using Thorpe-Ziegler cyclization. These substituted pyrroles are readily converted into 5H-pyrrolo[3,2-d] pyrimidine (9-deazapurines).
引用
收藏
页码：180 / 190
页数：11
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