SYNTHESIS OF CONDENSED PYRIMIDINES IN ONE-POT REACTION FROM PYRANOQUINOLINES AND BMMAs

被引:0
|
作者
Nahas, Nariman M. [1 ]
机构
[1] Umm Al Qura Univ, Dept Chem, Fac Sci Appl, Mecca, Saudi Arabia
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
New pentacyclic heterocycles of the type 3a-e -5a-e were synthesized by one - pot reaction of the amino-cyano pyrano[3,2-h]quinolines 1a-e with BMMAs (e.g. Ethyl N-[bis(methylsulfanyl) methylene] glycinate, ethyl 2[bis (methylsulfanyl) methylene]-1-methylhydrazine carboxylate and/or ethyl N[bis(methylsulfanyl) methylene]- beta-alaninate). All the synthesized derivatives were identified by conventional methods (IR, (HNMR)-H-1, MS) and elemental analysis. Antifungal tests were also performed.
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页码:51 / 54
页数:4
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