Copper-catalyzed cross-dehydrogenative coupling between quinazoline-3-oxides and indoles

被引：13
|
作者：
Yang, Qin [1 ]
Yin, Zhijian [1 ]
Zheng, Lifang [1 ]
Yuan, Jianjun [1 ]
Wei, Song [1 ]
Ding, Qiuping [1 ]
Peng, Yiyuan [1 ]
机构：
[1] Jiangxi Normal Univ, Jiangxi Prov Key Lab Green Chem, Minist Educ, Key Lab Funct Small Organ Mol, Nanchang 330022, Jiangxi, Peoples R China
来源：
RSC ADVANCES | 2019年 / 9卷 / 11期
基金：
中国国家自然科学基金;
关键词：
QUINOLINE N-OXIDES; C-H ARYLATION; ONE-STEP CONVERSION; EFFICIENT ROUTE; FUNCTIONALIZATION; ACTIVATION; ARYL; QUINAZOLINE-4-TOSYLATES; ELECTROLUMINESCENT; AZAAROMATICS;
D O I：
10.1039/c8ra09864f
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A novel and simple protocol for the synthesis of 4-(indole-3-yl)quinazolines via cross-dehydrogenative coupling of quinazoline-3-oxides and indoles under an air atmosphere has been developed. A series of biheteroaryl products were obtained in moderate to good yields.
引用
收藏
页码：5870 / 5877
页数：8
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