Copper-catalyzed cross-dehydrogenative coupling between quinazoline-3-oxides and indoles

被引：13

作者：

Yang, Qin ^{[1
]}

Yin, Zhijian ^{[1
]}

Zheng, Lifang ^{[1
]}

Yuan, Jianjun ^{[1
]}

Wei, Song ^{[1
]}

Ding, Qiuping ^{[1
]}

Peng, Yiyuan ^{[1
]}

机构：

[1] Jiangxi Normal Univ, Jiangxi Prov Key Lab Green Chem, Minist Educ, Key Lab Funct Small Organ Mol, Nanchang 330022, Jiangxi, Peoples R China

来源：

RSC ADVANCES | 2019年 / 9卷 / 11期

基金：

中国国家自然科学基金;

关键词：

QUINOLINE N-OXIDES; C-H ARYLATION; ONE-STEP CONVERSION; EFFICIENT ROUTE; FUNCTIONALIZATION; ACTIVATION; ARYL; QUINAZOLINE-4-TOSYLATES; ELECTROLUMINESCENT; AZAAROMATICS;

D O I：

10.1039/c8ra09864f

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A novel and simple protocol for the synthesis of 4-(indole-3-yl)quinazolines via cross-dehydrogenative coupling of quinazoline-3-oxides and indoles under an air atmosphere has been developed. A series of biheteroaryl products were obtained in moderate to good yields.

引用

页码：5870 / 5877

页数：8

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