Discovery of triazolopyridines as potent and selective acyl-CoA: Diacylglycerol acyltranferase 1 (DGAT1) inhibitors

被引:0
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作者
Sun, Chongqing [1 ]
Huang, Yanting [1 ]
Tuerdi, Huji [2 ]
Chao, Hannguang [2 ]
Peterson, Tara [3 ]
Dong, Jessica [3 ]
Chu, Ching-Hsuen [3 ]
Ma, Zhengping [3 ]
Chen, Luping [3 ]
Seethala, Ramakrishna [3 ]
Harvey, Susan [3 ]
Godonis, Helen [3 ]
Rooney, Suzanne [3 ]
Devenny, James [3 ]
Pelleymounter, Maryann [3 ]
Cai, Hong [4 ]
Fura, Aberra [4 ]
Ewing, William [1 ]
Poss, Michael [2 ]
Cheng, Dong [3 ]
Lawrence, R. Michael [2 ]
机构
[1] Bristol Myers Squibb Co, Metab Dis, New York, NY 10154 USA
[2] Bristol Myers Squibb Co, Early Discovery Chem, New York, NY 10154 USA
[3] Bristol Myers Squibb Co, Metab Dis Biol, New York, NY 10154 USA
[4] Bristol Myers Squibb Co, Preclin Candidate Optimizat, New York, NY 10154 USA
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
418-MEDI
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页数:1
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