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- [42] Synthesis and biological evaluation of 3,6-disubstituted [1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives as a novel class of potential anti-tumor agentsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2009, 44 (07) : 2776 - 2781Ibrahim, D. A.论文数: 0 引用数: 0 h-index: 0机构: Natl Org Drug Control & Res, Cairo 111321, Gizaa, Egypt Natl Org Drug Control & Res, Cairo 111321, Gizaa, Egypt
- [43] Discovery of JNJ-88549968, a Novel, First-in-Class CALRmutxCD3 T-Cell Redirecting Antibody for the Treatment of Myeloproliferative NeoplasmsBLOOD, 2023, 142Kuchnio, Anna论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumSamakai, Elsie论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Spring House, PA USA Janssen Res & Dev, Beerse, BelgiumHug, Eva论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumBalmana, Meritxell论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumJanssen, Lut论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumAmorim, Ricardo论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumCornelissen, Ivo论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumMajoros, Andrea论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumBroux, Michael论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumTaneja, Isha论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Spring House, PA USA Janssen Res & Dev, Beerse, BelgiumTorti, Vince论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, La Jolla, CA USA Janssen Res & Dev, Beerse, BelgiumAgic, Azra论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumMoritsch, Stefan论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumBenedetti, Filippo论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumRosebrock, Felix论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumPackman, Kathryn论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Cambridge, MA USA Janssen Res & Dev, Beerse, BelgiumArts, Janine论文数: 0 引用数: 0 h-index: 0机构: Janssen Sci Innovat Oncol, Beerse, Belgium Janssen Res & Dev, Beerse, BelgiumPatel, Sonal论文数: 0 引用数: 0 h-index: 0机构: Janssen Sci Innovat Oncol, London, England Janssen Res & Dev, Beerse, BelgiumLomas, Oliver Christopher论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, High Wycombe, England Janssen Res & Dev, Beerse, BelgiumDeyoung, M. Phillip论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Spring House, PA USA Janssen Res & Dev, Beerse, BelgiumZagrijtschuk, Oleh论文数: 0 引用数: 0 h-index: 0机构: MyeloPro Diagnost & Res GmbH, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumElsayed, Yusri论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Spring House, PA USA Janssen Res & Dev, Beerse, BelgiumConstantinescu, Stefan论文数: 0 引用数: 0 h-index: 0机构: Ludwig Inst Canc Res, Brussels, Belgium UCLouvain, Duve Inst, Brussels, Belgium Wel Res Inst, Welbio Dept, Wavre, Belgium Univ Oxford, Nuffield Dept Med, Ludwig Canc Res Oxford, Oxford, England Janssen Res & Dev, Beerse, BelgiumKralovics, Robert论文数: 0 引用数: 0 h-index: 0机构: Med Univ Vienna, Vienna, Austria Janssen Res & Dev, Beerse, BelgiumPhilippar, Ulrike论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev LLC, Beerse, Belgium Janssen Res & Dev, Beerse, Belgium
- [44] Discovery of 3-Substituted 1H-Indole-2-carboxylic Acid Derivatives as a Novel Class of CysLT1 Selective AntagonistsACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (03): : 335 - 339Chen, Huayan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaYang, Hui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaWang, Zhilong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaXie, Xin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R ChinaNan, Fajun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Natl Ctr Drug Screening, State Key Lab Drug Res, Shanghai 201203, Peoples R China
- [45] Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (09) : 2229 - 2250Kojima, Takuto论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanMochizuki, Michiyo论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanTakai, Takafumi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanHoashi, Yasutaka论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanMorimoto, Sachie论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanSeto, Masaki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanNakamura, Minoru论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanKobayashi, Katsumi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan ChromaJean Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanSako, Yuu论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanTanaka, Maiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanKanzaki, Naoyuki论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Seedsupply Ltd, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanKosugi, Yohei论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanYano, Takahiko论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Taisho Pharmaceut Co Ltd, Kita Ku, 403,Yoshino Cho 1 Chome, Saitama, Saitama 3319530, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, JapanAso, Kazuyoshi论文数: 0 引用数: 0 h-index: 0机构: Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Axcelead Drug Discovery Partners Inc, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan Takeda Pharmaceut Co Ltd, Res Div, 26-1,Muraoka Higashi 2 Chome, Fujisawa, Kanagawa 2510012, Japan
- [46] Discovery of 1,2,4-oxadiazole derivatives as a novel class of noncompetitive inhibitors of 3-hydroxykynurenine transaminase (HKT) from Aedes aegyptiBIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (02)Maciel, Larissa G.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilOliveira, Andrew A.论文数: 0 引用数: 0 h-index: 0机构: Univ Sao Paulo, Sao Carlos Inst Phys, Ave Joao Dagnone,1100 Jardim Santa Angelina, BR-13563120 Sao Carlos, SP, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilRomao, Tatiany P.论文数: 0 引用数: 0 h-index: 0机构: Fiocruz MS, IAM, Ave Prof Moraes Rego S-N, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilLeal, Laylla L. L.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilGuido, Rafael V. C.论文数: 0 引用数: 0 h-index: 0机构: Univ Sao Paulo, Sao Carlos Inst Phys, Ave Joao Dagnone,1100 Jardim Santa Angelina, BR-13563120 Sao Carlos, SP, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilSilva-Filha, Maria Helena N. L.论文数: 0 引用数: 0 h-index: 0机构: Fiocruz MS, IAM, Ave Prof Moraes Rego S-N, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazildos Anjos, Janaina V.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, BrazilSoares, Thereza A.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazil Univ Fed Pernambuco, Dept Fundamental Chem, Ave Jornalista Anibal Fernandes S-N Cidade Univ, BR-50740560 Recife, PE, Brazil
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