Synthesis and Phytotoxic Activity of 1,2,3-Triazole Derivatives

被引：58

作者：

Borgati, Thiago F. ^{[1
]}

Alves, Rosemeire B. ^{[1
]}

Teixeira, Robson R. ^{[2
]}

de Freitas, Rossimiriam P. ^{[2
]}

Perdigao, Thays G. ^{[2
]}

da Silva, Silma F. ^{[2
]}

dos Santos, Aline Aparecida ^{[2
]}

Bastidas, Alberto de Jesus O. ^{[3
]}

机构：

[1] Univ Fed Minas Gerais, Dept Quim, BR-31270900 Belo Horizonte, MG, Brazil

[2] Univ Fed Vicosa, Dept Quim, BR-36570000 Vicosa, MG, Brazil

[3] Nucleo Univ Pedro Rincon Gutierrez, Univ Los Andes, Fac Ciencias, Lab Quim Ecol,Dept Quim, Merida 5101 A, Venezuela

来源：

JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY | 2013年 / 24卷 / 06期

关键词：

herbicides; 1,2,3-triazoles; click chemistry; phytotoxicity; HERBICIDES; ALLELOCHEMICALS; DEGRADATION; PRODUCTS;

D O I：

10.5935/0103-5053.20130121

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Thirteen triazole derivatives bearing halogenated benzyl substituents were synthesized using the Cu-catalyzed azide-alkyne cycloaddition (CuAAC), a leading example of the click chemistry approach, as the key step. The biological activity of the compounds was evaluated, and it was found that these compounds interfere with the germination and radicle growth (shoots and roots) of two dicotyledonous species, Lactuca sativa and Cucumis sativus, and one monocotyledonous species, Allium cepa. The compounds showed predominantly inhibitory activity related to the evaluated species mainly at the concentration of 10(-4) mol L-1. Some of them presented inhibitory activity comparable to 2,4-D (2,4-dichlorophenoxyacetic acid), used as positive control.

引用

页码：953 / U805

页数：72

共 50 条

[1] Synthesis of Tyrosol 1,2,3-Triazole Derivatives and Their Phytotoxic Activity against Euphorbia heterophylla
Franco, Cristiane Aparecida
da Silva, Toshik Iarley
Dias, Marlon Gomes
Ferreira, Bruno Wesley
de Sousa, Bianca Lana
Bousada, Guilherme Mateus
Barreto, Robert Weingart
Vaz, Boniek Gontijo
Lima, Gesiane da Silva
Santos, Marcelo Henrique dos
Grossi, Jose Antonio Saraiva
Varejao, Eduardo Vinicius Vieira
[J]. JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2022, 70 (09) : 2806 - 2816
[2] SYNTHESIS OF 1,2,3-TRIAZOLE DERIVATIVES
CARBONI, S
DASETTIMO, A
FERRARINI, PL
LIVI, O
TONETTI, I
[J]. CHIMICA & L INDUSTRIA, 1976, 58 (12): : 878 - 878
[3] Synthesis of 1,2,3-Triazole Derivatives
Jiang Yubo
Kuang Chunxiang
[J]. PROGRESS IN CHEMISTRY, 2012, 24 (10) : 1983 - 1994
[4] SYNTHESIS AND CYTOTOXIC ACTIVITY OF 1,2,3-TRIAZOLE DERIVATIVES OF EUGENOL
Rodrigues Gazolla, Poliana Aparecida
Teixeira, Robson Ricardo
da Silva, Adalberto Manoel
Vaz, Boniek Gontijo
Vasconcelos, Gessica Adriana
Siqueira, Raoni Pais
Sousa Goncalves, Victor Hugo
Pereira, Higor Sette
Bressan, Gustavo Costa
[J]. QUIMICA NOVA, 2018, 41 (05): : 497 - 506
[5] Synthesis and antifungal activity of 1,2,3-triazole phenylhydrazone derivatives
Dai, Zhi-Cheng
Chen, Yong-Fei
Zhang, Mao
Li, Sheng-Kun
Yang, Ting-Ting
Shen, Li
Wang, Jian-Xin
Qian, Shao-Song
Zhu, Hai-Liang
Ye, Yong-Hao
[J]. ORGANIC & BIOMOLECULAR CHEMISTRY, 2015, 13 (02) : 477 - 486
[6] SYNTHESIS AND HERBICIDAL ACTIVITY OF NOVEL 1,2,3-TRIAZOLE DERIVATIVES
GOH, A
USUI, Y
HAYASHIZAKI, K
TSUTSUMI, Y
TAMURA, K
YAMADA, S
[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1994, 207 : 67 - AGRO
[7] Synthesis of glucosylated 1,2,3-triazole derivatives
Chen, XM
Li, ZJ
Ren, ZX
Huang, ZT
[J]. CARBOHYDRATE RESEARCH, 1999, 315 (3-4) : 262 - 267
[8] HERBICIDAL ACTIVITY OF 1,2,3-TRIAZOLE DERIVATIVES
MESSORI, V
BALDI, L
BIANCHETTI, G
[J]. CHIMICA & L INDUSTRIA, 1977, 59 (06): : 438 - 440
[9] Synthesis of ribosylated 1,2,3-triazole derivatives
Ren, ZX
Chen, XM
Li, ZJ
Huang, ZT
[J]. HETEROATOM CHEMISTRY, 2003, 14 (06) : 487 - 490
[10] Synthesis of glucosylated 1,2,3-triazole derivatives
[J]. Carbohyd Res, 3-4 (262-267):

← 1 2 3 4 5 →