Convenient Synthesis of Benzoxazolone Derivatives by Cross-Coupling of Benzoxazolone Boronates with Aryl Halides

被引：0

作者：

Fukaya, Takayuki ^{[1
]}

Masumoto, Shuji ^{[1
]}

机构：

[1] Dainippon Sumitomo Pharma Co Ltd, Drug Res Div, Suita, Osaka 5640053, Japan

来源：

SYNTHESIS-STUTTGART | 2013年 / 45卷 / 23期

关键词：

heterocycles; boron; cross-coupling; biaryls; catalysis; arylations; LIGANDS; DESIGN; ESTERS;

D O I：

10.1055/s-0033-1339799

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Benzoxazolone derivatives with various substituents at the C-5 position were synthesized efficiently via benzoxazolone boronates as the key intermediate. The target compounds were also synthesized from (het)aryl halides in a one-pot process. These methods permitted efficient exploratory syntheses of a series of benzoxazolone derivatives.

引用

页码：3269 / 3275

页数：7

共 50 条

[21] PALLADIUM-CATALYZED CROSS-COUPLING REACTION OF HETEROARYLTRIOLBORATES WITH ARYL HALIDES FOR SYNTHESIS OF BIARYLS
Yamamoto, Yasunori
Takizawa, Miho
Yu, Xiao-Qiang
Miyaura, Norio
HETEROCYCLES, 2010, 80 (01) : 359 - 368
[22] Stilbene synthesis through decarboxylative cross-coupling of substituted cinnamic acids with aryl halides
Rameau, Nelly
Russo, Baptiste
Mangematin, Stephane
Pinel, Catherine
Djakovitch, Laurent
APPLIED CATALYSIS A-GENERAL, 2018, 560 : 132 - 143
[23] Synthesis of unsymmetrical biaryls by electroreductive cobalt-catalyzed cross-coupling of aryl halides
Gomes, P
Fillon, H
Gosmini, C
Labbé, E
Périchon, J
TETRAHEDRON, 2002, 58 (42) : 8417 - 8424
[24] SYNTHESIS AND IN-VITRO ACTIVITY OF NEW CEPHEM DERIVATIVES WITH BENZOXAZOLONE RING
MINCHEVA, ZP
KALCHEVA, VB
GOLOVINSKY, EG
TABAKOVA, SV
PHARMAZIE, 1993, 48 (11): : 859 - 860
[25] Nickel-Catalyzed Reductive Cross-Coupling of Aryl Halides
Qian, Qun
Zang, Zhenhua
Wang, Shulin
Chen, Yang
Lin, Kunhua
Gong, Hegui
SYNLETT, 2013, 24 (05) : 619 - 624
[26] Enantioselective Cross-Coupling of meso-Epoxides with Aryl Halides
Zhao, Yang
Weix, Daniel J.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2015, 137 (09) : 3237 - 3240
[27] Cross-coupling of alkynylsilanols with aryl halides promoted by potassium trimethylsilanolate
Denmark, SE
Tymonko, SA
JOURNAL OF ORGANIC CHEMISTRY, 2003, 68 (23): : 9151 - 9154
[28] PALLADIUM-CATALYZED CROSS-COUPLING OF VINYLALANES WITH ARYL HALIDES
ALHASSAN, MI
SYNTHETIC COMMUNICATIONS, 1987, 17 (12) : 1413 - 1420
[29] Decarboxylative Cross-Coupling of Azoyl Carboxylic Acids with Aryl Halides
Zhang, Fengzhi
Greaney, Michael F.
ORGANIC LETTERS, 2010, 12 (21) : 4745 - 4747
[30] Cobalt-Catalyzed Cross-Coupling Reactions Aryl Halides
Gosmini, Corinne
Moncomble, Aurelien
ISRAEL JOURNAL OF CHEMISTRY, 2010, 50 (5-6) : 568 - 576

← 1 2 3 4 5 →