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- [1] Phase 1 Clinical Evaluation of the CCR2 Antagonist CCX872-BDIABETES, 2013, 62 : A292 - A293Bekker, Pirow论文数: 0 引用数: 0 h-index: 0Charvat, Trevor论文数: 0 引用数: 0 h-index: 0Miao, Shichang论文数: 0 引用数: 0 h-index: 0Lohr, Lisa论文数: 0 引用数: 0 h-index: 0Sullivan, Timothy论文数: 0 引用数: 0 h-index: 0Miao, Zhenhua论文数: 0 引用数: 0 h-index: 0Powers, Jay论文数: 0 引用数: 0 h-index: 0Jaen, Juan论文数: 0 引用数: 0 h-index: 0Schall, Thomas J.论文数: 0 引用数: 0 h-index: 0
- [2] Orally administered CCR2 selective inhibitor CCX872-b clinical trial in pancreatic cancer.JOURNAL OF CLINICAL ONCOLOGY, 2017, 35 (04)Noel, Marcus Smith论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAHezel, Aram F.论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USALinehan, David论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAWang-Gillam, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAEskens, Ferry论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USASleijfer, Stefan论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USADesar, Ingrid论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAErdkamp, Frans论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAWilmink, Johanna论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USADiehl, Janet论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAPotarca, Antonia论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAZhao, Niky论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USADeng, Jun论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USALohr, Lisa论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USAMiao, Shichang论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USACharo, Israel论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USASingh, Rajinder论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USASchall, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USABekker, Pirow论文数: 0 引用数: 0 h-index: 0机构: Univ Rochester, Med Ctr, Wilmot Canc Inst, Rochester, NY 14642 USA
- [3] CCR2 antagonist CCX140-B provides renal and glycemic benefits in diabetic transgenic human CCR2 knockin miceAMERICAN JOURNAL OF PHYSIOLOGY-RENAL PHYSIOLOGY, 2013, 305 (09) : F1288 - F1297Sullivan, Timothy论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAMiao, Zhenhua论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USADairaghi, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAKrasinski, Antoni论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAWang, Yu论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAZhao, Bin N.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USABaumgart, Trageen论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAErtl, Linda S.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAPennell, Andrew论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USASeitz, Lisa论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAPowers, Jay论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAZhao, Ruiping论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAUngashe, Solomon论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAWei, Zheng论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USABoring, Landin论文数: 0 引用数: 0 h-index: 0机构: J David Gladstone Res Inst, Gladstone Inst Cardiovasc Dis, San Francisco, CA USA ChemoCentryx Inc, Mountain View, CA USATsou, Chia-Lin论文数: 0 引用数: 0 h-index: 0机构: J David Gladstone Res Inst, Gladstone Inst Cardiovasc Dis, San Francisco, CA USA ChemoCentryx Inc, Mountain View, CA USACharo, Israel论文数: 0 引用数: 0 h-index: 0机构: J David Gladstone Res Inst, Gladstone Inst Cardiovasc Dis, San Francisco, CA USA ChemoCentryx Inc, Mountain View, CA USABerahovich, Robert D.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USASchall, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAJaen, Juan C.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USA
- [4] The inhibition of CCR2 to modify the microenvironment in pancreatic cancer mouse model and to support the profiling of the CCR2 inhibitor CCX872-B in patients.JOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (15)Wang-Gillam, Andrea论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USANoel, Marcus Smith论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USASleijfer, Stefan论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USAJung, Heiyoun论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USALohr, Lisa论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USAZhao, Niky论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USAMiao, Shichang论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USAPotarca, Antonia论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USACharo, Israel论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USABekker, Petrus论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USASchall, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Siteman Canc Ctr, St Louis, MO USA
- [5] The effect of CCR2 inhibitor CCX140-B on residual albuminuria in patients with type 2 diabetes and nephropathy: a randomised trialLANCET DIABETES & ENDOCRINOLOGY, 2015, 3 (09): : 687 - 696de Zeeuw, Dick论文数: 0 引用数: 0 h-index: 0机构: Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, Netherlands Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsBekker, Pirow论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsHenkel, Elena论文数: 0 引用数: 0 h-index: 0机构: Tech Univ Dresden, Ctr Clin Studies, D-01062 Dresden, Germany Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsHasslacher, Christopher论文数: 0 引用数: 0 h-index: 0机构: Inst Diabet Endocrinol & Metab Dis, Heidelberg, Germany Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsGouni-Berthold, Ioanna论文数: 0 引用数: 0 h-index: 0机构: Univ Cologne, Ctr Endocrinol Diabet & Prevent Med, D-50931 Cologne, Germany Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsMehling, Heidrun论文数: 0 引用数: 0 h-index: 0机构: Charite Expt & Clin Res Ctr, Berlin, Germany Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsPotarca, Antonia论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsTesar, Vladimir论文数: 0 引用数: 0 h-index: 0机构: Charles Univ Prague, Sch Med 1, Dept Nephrol, Prague, Czech Republic Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsHeerspink, Hiddo J. Lambers论文数: 0 引用数: 0 h-index: 0机构: Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, Netherlands Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, NetherlandsSchall, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA Univ Groningen, Univ Med Ctr Groningen, Dept Clin Pharm & Pharmacol, Groningen, Netherlands
- [6] Chemokine receptor 2 antagonist CCX140-B in Phase 2 for type 2 diabetesDIABETOLOGIA, 2010, 53Sullivan, T.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAMiao, S.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USABerahovich, R.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAZhao, N.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAUngashe, S.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAJohnson, D.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USABekker, P.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAJean, J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USASchall, T. J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USA
- [7] CCR2 INHIBITOR CCX140 EFFECTIVE IN PHASE 2 CLINICAL TRIAL IN DIABETIC NEPHROPATHYNEPHROLOGY DIALYSIS TRANSPLANTATION, 2015, 30de Zeeuw, Dick论文数: 0 引用数: 0 h-index: 0机构: Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, Netherlands Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsHenkel, Elena论文数: 0 引用数: 0 h-index: 0机构: Tech Univ Dresden, Diabet, D-01062 Dresden, Germany Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsPsottova, Jana论文数: 0 引用数: 0 h-index: 0机构: Diainmed, Diabet, Prague, Czech Republic Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, Netherlands论文数: 引用数: h-index:机构:Mehling, Heidrun论文数: 0 引用数: 0 h-index: 0机构: Free Univ Berlin, Diabet, Berlin, Germany Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsHasslacher, Christopher论文数: 0 引用数: 0 h-index: 0机构: Heidelberg Univ, Diabet, Heidelberg, Germany Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsPotarca, Antonia论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Clin Operat, Mountain View, CA USA Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsBekker, Pirow论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Med & Clin Affairs, Mountain View, CA USA Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, NetherlandsSchall, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, R&D, Mountain View, CA USA Univ Med Ctr Groningen, Clin Pharm & Pharmacol, NL-9713 AV Groningen, Netherlands
- [8] Reduction of Liver Fibrosis by CCR2 antagonist CCX872 in Murine Models of NASHHEPATOLOGY, 2016, 64 : 763A - 763AMiao, Zhenhua论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USANewland, Dale论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USAErtl, Linda论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USAParker, Richard论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Birmingham NHS Fdn Trust, Birmingham, W Midlands, England ChemoCentryx, Mountain View, CA USAMcMahon, Jeff论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USAZhang, Penglie论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USAAdams, David H.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Birmingham NHS Fdn Trust, Birmingham, W Midlands, England ChemoCentryx, Mountain View, CA USAScholl, Thomas J.论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USACharo, Israel论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx, Mountain View, CA USA ChemoCentryx, Mountain View, CA USA
- [9] Therapeutic use of a clinical stage CCR2 inhibitor, CCX872, in obesity-associated steatohepatitisLANCET, 2014, 383 : 78 - 78Parker, Richard论文数: 0 引用数: 0 h-index: 0机构: Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, England ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandWalters, Matthew论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandErtl, Linda论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandEbsworth, Karen论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandTan, Joanne论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandMcMahon, Jeff论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandPowers, Jay论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandAdams, David论文数: 0 引用数: 0 h-index: 0机构: Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, England Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandJaen, Juan论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, EnglandSchall, Tom论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA Univ Birmingham, Liver Res Ctr, Birmingham B15 2TT, W Midlands, England
- [10] Reduction of Liver Fibrosis by CCR2 Antagonist CCX872 in Murine Models of NASHAMERICAN JOURNAL OF GASTROENTEROLOGY, 2016, 111 : S398 - S398Miao, Zhenhua论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USANewland, Dale论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAErtl, Linda论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USA论文数: 引用数: h-index:机构:McMahon, Jeff论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USAZhang, Penglie论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USA论文数: 引用数: h-index:机构:Schall, Thomas论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USACharo, Israel论文数: 0 引用数: 0 h-index: 0机构: ChemoCentryx Inc, Mountain View, CA USA ChemoCentryx Inc, Mountain View, CA USA