Synthesis of new methyl derivatives of aza- and diazaphenanthrene

被引:9
|
作者
Kozlov, N. G. [1 ]
Gusak, K. N. [1 ]
机构
[1] Natl Acad Sci Belarus, Inst Phys Organ Chem, Minsk 220072, BELARUS
关键词
Quinoline; Methyl Derivative; Methyl Vinyl Ketone; Aminoketone; Intermediate Reaction Product;
D O I
10.1134/S1070428008070178
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
By condensation of acetone with 2-naphthylamine and 3-(4-fluorophenyl)-1H-pyrazole-4-, pyridine-3-, quinoline-2-, quinoline-6-carbaldehyde and 4-(2-fluorobenzyloxy) benzaldehyde new 3-aryl(heteryl)-1-methylbenzo[f]quinolines were synthesized. Reactions of acetone with 6-quinolylamine and aromatic aldehydes provided 3-aryl-1-methyl-4,7-phenanthrolines. Intermediate reaction products were isolated: 4- phenyl-or (3-pyridyl)-4-(2-naphthylamino or 6-quinolylamino)butan-2-ones.
引用
收藏
页码:1049 / 1053
页数:5
相关论文
共 50 条
  • [31] Synthesis of new C-glycosyl aza-β3-amino acids building blocks
    Andreini, Manuel
    Felten, Anne-Sophie
    Thien, Hoang-Trang Tran
    Taillefumier, Claude
    Pellegrini-Moise, Nadia
    Chapleur, Yves
    TETRAHEDRON LETTERS, 2012, 53 (22) : 2702 - 2705
  • [32] Synthesis of α,α-disubstituted unnatural amino acid derivatives using the aza-[2,3]-Wittig sigmatropic rearrangement
    Anderson, JC
    Skerratt, S
    JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 2002, (24): : 2871 - 2879
  • [33] An aerobic oxidative aza-[4+2] cycloaddition induced by radical cation salt: Synthesis of dihydroquinazoline derivatives
    Luo, Liangliang
    Zhao, Xiaolong
    Zhang, Liang
    Yuan, Yu
    Lu, Shiwei
    Jia, Xiaodong
    TETRAHEDRON LETTERS, 2016, 57 (51) : 5830 - 5833
  • [34] Aza-β3-cyclotetrapeptides
    Salauen, Arnaud
    Mocquet, Clemence
    Perochon, Romain
    Lecorgne, Aurelien
    Le Grel, Barbara
    Potel, Michel
    Le Grel, Philippe
    JOURNAL OF ORGANIC CHEMISTRY, 2008, 73 (21): : 8579 - 8582
  • [35] New functionalized aza-β3-aminoacids for click chemistry
    Abbour, S.
    Mosbah, A.
    Baudy-Floc'h, M.
    JOURNAL OF PEPTIDE SCIENCE, 2012, 18 : S183 - S184
  • [36] Palladium-catalyzed amination in the synthesis of aza- and diazacrown trismacrocyclic compounds
    Yakushev, A. A.
    Anokhin, M. V.
    Averin, A. D.
    Maloshitskaya, O. A.
    Beletskaya, I. P.
    RUSSIAN CHEMICAL BULLETIN, 2012, 61 (07) : 1474 - 1482
  • [37] Organocatalytic enantioselective synthesis of acyclic pyrimidine nucleosides by aza- Michael reaction
    Lee, Su-Jeong
    Ahn, Jun-Gi
    Seo, Jihwan
    Ha, Heun-Jong
    Cho, Chang-Woo
    ORGANIC & BIOMOLECULAR CHEMISTRY, 2018, 16 (48) : 9477 - 9486
  • [38] Palladium-catalyzed amination in the synthesis of aza- and diazacrown trismacrocyclic compounds
    A. A. Yakushev
    M. V. Anokhin
    A. D. Averin
    O. A. Maloshitskaya
    I. P. Beletskaya
    Russian Chemical Bulletin, 2012, 61 : 1474 - 1482
  • [39] Modular Synthesis of Bicyclic and Tricyclic (Aza-) Arenes from Nucleophilic (Aza-)Arenes with Electrophilic Side Arms via [4+2] Annulation Reactions
    Huang, Wenbo
    Chen, Shaomin
    Yang, Jian
    El-Harairy, Ahmed
    Wang, Xin
    Li, Minghao
    Gu, Yanlong
    ADVANCED SYNTHESIS & CATALYSIS, 2019, 361 (18) : 4369 - 4378
  • [40] New Building Blocks for Solid-Phase Synthesis of Peptide Analogues: Nβ-Fmoc-Nβ-Methyl- aza-β3-amino acides
    Baudy-Floc'h, D. R.
    Kisselnova, K.
    Nicolas, I.
    Jaerv, J.
    Bauchat, P.
    JOURNAL OF PEPTIDE SCIENCE, 2010, 16 : 58 - 59