Facile Preparation of Indoles and 1,2-Benzothiazine 1,1-Dioxides: Nucleophilic Addition of Sulfonamides to Bromoacetylenes and Subsequent Palladium-Catalyzed Cyclization

被引：49
|
作者：
Yamagishi, Masahito [1 ]
Nishigai, Ken [1 ]
Ishii, Azusa [1 ]
Hata, Takeshi [1 ]
Urabe, Hirokazu [1 ]
机构：
[1] Tokyo Inst Technol, Grad Sch Biosci & Biotechnol, Dept Biomol Engn, Midori Ku, Yokohama, Kanagawa 2268501, Japan
来源：
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION | 2012年 / 51卷 / 26期
关键词：
alkynes; cyclizations; indoles; nucleophilic addition; palladium; DIRECT ARYLATION; ALKYNES; DEPROTECTION; IMIDAZOLES; MECHANISM; ANILINES; BROMIDES; ACCESS;
D O I：
10.1002/anie.201201024
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
75
引用
收藏
页码：6471 / 6474
页数：4
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