Facile Preparation of Indoles and 1,2-Benzothiazine 1,1-Dioxides: Nucleophilic Addition of Sulfonamides to Bromoacetylenes and Subsequent Palladium-Catalyzed Cyclization

被引：49

作者：

Yamagishi, Masahito ^{[1
]}

Nishigai, Ken ^{[1
]}

Ishii, Azusa ^{[1
]}

Hata, Takeshi ^{[1
]}

Urabe, Hirokazu ^{[1
]}

机构：

[1] Tokyo Inst Technol, Grad Sch Biosci & Biotechnol, Dept Biomol Engn, Midori Ku, Yokohama, Kanagawa 2268501, Japan

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION | 2012年 / 51卷 / 26期

关键词：

alkynes; cyclizations; indoles; nucleophilic addition; palladium; DIRECT ARYLATION; ALKYNES; DEPROTECTION; IMIDAZOLES; MECHANISM; ANILINES; BROMIDES; ACCESS;

D O I：

10.1002/anie.201201024

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

引用

页码：6471 / 6474

页数：4

共 33 条

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[6] Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation of Thietane 1,1-Dioxides
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ORGANIC LETTERS, 2022, 24 (01) : 400 - 405
[7] 3-ACYL-4-HYDROXY-2H-1,2-BENZOTHIAZINE 1,1-DIOXIDES .1. ALKYLATION, AMINATION, AND ETHOXYCARBONYLATION
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[8] C-13 NMR ANALYSIS OF SOME 4-HYDROXY-2H-1,2-BENZOTHIAZINE 1,1-DIOXIDES
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PERILLO, IA
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1993, 30 (04) : 1051 - 1056
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CHINESE CHEMICAL LETTERS, 1996, 7 (12) : 1073 - 1076
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