Protein farnesyltransferase inhibitors exhibit potent anti-malarial activity.

被引:0
|
作者
Nallan, L
Bauer, K
Bendale, PM
Yokayama, K
Hucke, O
Verlinde, CLMJ
Floyd, D
Lombardo, LJ
Williams, D
Van Voorhis, WC
Gelb, MH
机构
[1] Univ Washington, Dept Chem, Seattle, WA 98195 USA
[2] Univ Washington, Dept Med, Seattle, WA USA
[3] Univ Washington, Dept Biochem, Seattle, WA 98195 USA
[4] Univ Washington, Biomol Struct Ctr, Seattle, WA USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
383-MEDI
引用
收藏
页码:U177 / U177
页数:1
相关论文
共 50 条
  • [42] In vitro and in vivo assessment of the anti-malarial activity of Caesalpinia pluviosa
    Kayano, Ana Carolina A. V.
    Lopes, Stefanie C. P.
    Bueno, Fernanda G.
    Cabral, Elaine C.
    Souza-Neiras, Wanessa C.
    Yamauchi, Lucy M.
    Foglio, Mary A.
    Eberlin, Marcos N.
    Mello, Joao Carlos P.
    Costa, Fabio T. M.
    MALARIA JOURNAL, 2011, 10
  • [43] The Biological and Clinical Activity of Anti-Malarial Drugs In Autoimmune Disorders
    Taherian, Elham
    Rao, Anshul
    Malemud, Charles J.
    Askari, Ali D.
    CURRENT RHEUMATOLOGY REVIEWS, 2013, 9 (01) : 45 - 62
  • [44] ANTI-MALARIAL ACTIVITY IN ANIMALS OF THE OPTICAL ISOMERS OF CHLOROQUINE DIPHOSPHATE
    HABERKORN, A
    KRAFT, HP
    BLASCHKE, G
    TROPENMEDIZIN UND PARASITOLOGIE, 1979, 30 (03): : 308 - 312
  • [45] Prediction of Anti-Malarial Activity Based on Deep Belief Network
    Tian, Shengwei
    Yan, Yilin
    Yu, Long
    Wang, Mei
    Li, Li
    INTERNATIONAL JOURNAL OF COMPUTATIONAL INTELLIGENCE AND APPLICATIONS, 2018, 17 (03)
  • [46] ASPARAGINE ETHYLENEDIAMINES AS ANTI-MALARIAL PLASMODIUM-SELECTIVE PROTEASOME INHIBITORS
    Zhan, Wenhu
    Visone, Joeseph
    Harris, Jacob
    Ouellette, Tierra
    Wang, Rong
    Zang, Hao
    Singh, Pradeep
    Ginn, John
    Sukenick, George
    Wong, Tzu-Tshin
    Okoro, Judith
    Scales, Ryan
    Tumwebaze, Patrick K.
    Rosenthal, Philip J.
    Kafsack, Bjorn
    Cooper, Roland A.
    Meinke, Peter T.
    Lin, Gang
    Kirkman, Laura
    AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 2019, 101 : 2 - 2
  • [47] Imidazopyridazine analogues as anti-malarial PfPI3K inhibitors
    Liu, Rui
    Pandharkar, Trupti
    Safeukui, Innocent
    Bhattacharjee, Souvik
    Liu, Haining
    Wiest, Olaf
    Haldar, Kasturi
    Miller, Marvin
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 255
  • [48] Anti-malarial activity of geldanamycin derivatives in mice infected with Plasmodiumyoelii
    Rubul Mout
    Zhi-Dong Xu
    Angela K H Wolf
    Vincent Jo Davisson
    Gotam K Jarori
    Malaria Journal, 11
  • [49] Structurally novel, potent and selective inhibitors of protein farnesyltransferase.
    Yang, BWV
    Thompson, CB
    Kane, J
    Lyssikatos, JP
    Phillips, VV
    Paillet, S
    Tsaparikos, K
    Obach, RS
    Hagen, AE
    Kajiji, SM
    CLINICAL CANCER RESEARCH, 2000, 6 : 4494S - 4495S
  • [50] QSAR Models for Anti-Malarial Activity of 4-Aminoquinolines
    Masand, Vijay H.
    Toropov, Andrey A.
    Toropova, Alla P.
    Mahajan, Devidas T.
    CURRENT COMPUTER-AIDED DRUG DESIGN, 2014, 10 (01) : 75 - 82