Synthesis and evaluation of phosphonopeptide cathepsin C inhibitors

被引：0
|
作者：
Kafarski, P
Drag, M
Pawelczak, M
Berlicki, L
机构：
[1] Wroclaw Tech Univ, Inst Organ Chem Biochem & Biotechnol, PL-50370 Wroclaw, Poland
[2] Univ Opole, Inst Chem, PL-45052 Opole, Poland
来源：
BIOPOLYMERS | 2003年 / 71卷 / 03期
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
P431
引用
收藏
页码：396 / 396
页数：1
相关论文
共 50 条
  • [21] Design, synthesis, and biological evaluation of potent thiosemicarbazone based cathepsin L inhibitors
    Kumar, G. D. Kishore
    Chavarria, Gustavo E.
    Charlton-Sevcik, Amanda K.
    Arispe, Wara M.
    MacDonough, Matthew T.
    Strecker, Tracy E.
    Chen, Shen-En
    Siim, Bronwyn G.
    Chaplin, David J.
    Trawick, Mary Lynn
    Pinney, Kevin G.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (04) : 1415 - 1419
  • [22] Design, synthesis, and evaluation of inhibitors of cathepsin L: Exploiting a unique thiocarbazate chemotype
    Myers, Michael C.
    Shah, Parag P.
    Beavers, Mary Pat
    Napper, Andrew D.
    Diamond, Scott L.
    Smith, Amos B., III
    Huryn, Donna M.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (12) : 3646 - 3651
  • [23] Asymmetric synthesis and evaluation of epoxy-α-acyloxycarboxamides as selective inhibitors of cathepsin L
    dos Santos, Deborah A.
    Deobald, Anna Maria
    Cornelio, Vivian E.
    Avila, Roberta M. D.
    Cornea, Renata C.
    Bernasconi, Gilberto C. R.
    Paixao, Marcio W.
    Vieira, Paulo C.
    Correa, Arlene G.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (17) : 4620 - 4627
  • [24] Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C
    Guay, Daniel
    Beaulieu, Christian
    Reddy, T. Jagadeeswar
    Zamboni, Robert
    Methot, Nathalie
    Rubin, Joel
    Ethier, Diane
    Percival, M. David
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (18) : 5392 - 5396
  • [25] Design and synthesis of novel cathepsin C inhibitors with anti-inflammatory activity
    Shen, Xiaobao
    Li, Nan
    Liu, Miao
    Han, Xuanzheng
    Wang, Yazhi
    Jia, Jingwen
    Wu, Fufang
    Chen, Hongwei
    Liu, Xinhua
    RSC MEDICINAL CHEMISTRY, 2025, 16 (02): : 876 - 891
  • [26] Synthesis of novel phosphonopeptide derivatives and their biological activity
    Dai, Q
    Chen, RY
    HETEROATOM CHEMISTRY, 1997, 8 (03) : 279 - 282
  • [27] Development and evaluation of new cathepsin K inhibitors
    Tha, Soe
    Liang, Kenneth
    Obregon, Roxana
    Kadasala, Naveen Reddy
    Wen, Lisa
    Huang, Jenq Kuen
    McConnell, Rose
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241
  • [28] Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L
    Parker, Erica N.
    Song, Jiangli
    Kumar, G. D. Kishore
    Odutola, Samuel O.
    Chavarria, Gustavo E.
    Charlton-Sevcik, Amanda K.
    Strecker, Tracy E.
    Barnes, Ashleigh L.
    Sudhan, Dhivya R.
    Wittenborn, Thomas R.
    Siemann, Dietmar W.
    Horsman, Michael R.
    Chaplin, David J.
    Trawick, Mary Lynn
    Pinney, Kevin G.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (21) : 6974 - 6992
  • [29] Synthesis and evaluation of some semicarbazone- and thiosemicarbazone-based cathepsin B inhibitors
    Neera Raghav
    Ravinder Kaur
    Medicinal Chemistry Research, 2014, 23 : 4669 - 4679
  • [30] Synthesis and evaluation of new cathepsin D inhibitors containing substituted hydroxyethyl piperazine isosteres
    Velusamy, Priya
    Driver, Darryl
    Godwin, Walter E.
    McConnell, Rose M.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 233 : 528 - 528
12345