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- [21] Discovery of a novel and highly selective CDK9 kinase inhibitor (JS']JSH-009) with potent antitumor efficacy in preclinical acute myeloid leukemia modelsINVESTIGATIONAL NEW DRUGS, 2020, 38 (05) : 1272 - 1281Wang, Li论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaHu, Chen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Aoli论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaChen, Cheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWu, Jiaxin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaJiang, Zongru论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaZou, Fengming论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaYu, Kailin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Juan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wenliang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Zuowei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Beilei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaQi, Ziping论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Qingwang论文数: 0 引用数: 0 h-index: 0机构: Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaWang, Wenchao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLi, Lili论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Dept Hematol, Affiliated Hosp 1, Hefei 230022, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaGe, Jian论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Dept Hematol, Affiliated Hosp 1, Hefei 230022, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R ChinaLiu, Qingsong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China Univ Sci & Technol China, Hefei 230036, Anhui, Peoples R China Precis Med Res Lab Anhui Prov, Hefei 230088, Anhui, Peoples R China Chinese Acad Sci, Hefei Inst Phys Sci, Inst Technol Innovat, Precis Targeted Therapy Discovery Ctr, Hefei 230088, Anhui, Peoples R China Anhui Med Univ, Dept Hematol, Affiliated Hosp 1, Hefei 230022, Anhui, Peoples R China Anhui Univ, Inst Phys Sci & Informat Technol, Hefei 230601, Anhui, Peoples R China Chinese Acad Sci, High Field Magnet Lab, Key Lab High Magnet Field & Ion Beam Phys Biol, Hefei Inst Phys Sci, Mailbox 1110,350 Shushanhu Rd, Hefei 230031, Anhui, Peoples R China
- [22] OKI-1546 is a selective, orally bioavailable inhibitor of CDK12 that causes tumor regression in multiple preclinical cancer modelsCANCER RESEARCH, 2023, 83 (07)Strait, Alexander A.论文数: 0 引用数: 0 h-index: 0Mareska, David A.论文数: 0 引用数: 0 h-index: 0Mahadevan, Jyothi论文数: 0 引用数: 0 h-index: 0Schulte, Christie A.论文数: 0 引用数: 0 h-index: 0Izrayelit, Yevgeniy论文数: 0 引用数: 0 h-index: 0Boys, Mark L.论文数: 0 引用数: 0 h-index: 0Woessner, Richard论文数: 0 引用数: 0 h-index: 0
- [23] Pharmacological characterization of a preclinical candidate covalently inhibiting CDK12CANCER RESEARCH, 2019, 79 (13)Poddutoori, Ramulu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaRajagopalan, Sujatha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaMukherjee, Subhendu论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaMarappan, Sivapriya论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaSamiulla, D. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaSivakumar, Sasirekha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaNayak, Shilpa S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaRavindra, M., V论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaDevaraja, T. S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaKondela, Srinivas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaTgore, Suraj论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaDhudashiya, Amit A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaCharamanna, K. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaAravind, A. B.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaAmith, A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaPavithra, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaPathange, Hema Sankar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaAntony, Thomas论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaJaleel, Mahaboobi论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaGiri, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaDaginakatte, Girish论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaNellore, Kavitha论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaChelur, Shekar论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaRamachandra, Murali论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, IndiaSamajdar, Susanta论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Housr Rd, Bangalore, Karnataka, India
- [24] An oral and selective CDK12 inhibitor demonstrates robust anti-tumor activityCANCER RESEARCH, 2022, 82 (12)Hu, Shanhu论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMoebius, David论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USADworakowski, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACooper, Elliott论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USALaPlaca, Derek论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAAlnemy, Sydney论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAPerera, Phone论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMarineau, Jason论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAChuaqui, Claudio论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACarulli, John P.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOlson, Eric论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USA
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