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- [42] Targeting metabolic vulnerability in mitochondria conquers MEK inhibitor resistance in KRAS-mutant lung cancerACTA PHARMACEUTICA SINICA B, 2023, 13 (03) : 1145 - 1163Feng, Juanjuan论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China Southern Med Univ, Affiliated Fengxian Hosp, Joint Ctr Translat Med, Shanghai 201499, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaLian, Zhengke论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaXia, Xinting论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaLu, Yue论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaHu, Kewen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Shanghai Canc Ctr, Canc Inst, Shanghai Med Coll,Dept Oncol, Shanghai 200032, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaZhang, Yunpeng论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaLiu, Yanan论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaHu, Longmiao论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaYuan, Kun论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaSun, Zhenliang论文数: 0 引用数: 0 h-index: 0机构: Southern Med Univ, Affiliated Fengxian Hosp, Joint Ctr Translat Med, Shanghai 201499, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R ChinaPang, Xiufeng论文数: 0 引用数: 0 h-index: 0机构: East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China East China Normal Univ, Sch Life Sci, Shanghai Key Lab Regulatory Biol, Shanghai 200241, Peoples R China
- [43] KRAS Dimerization Impacts MEK Inhibitor Sensitivity and Oncogenic Activity of Mutant KRASCELL, 2018, 172 (04) : 857 - +Ambrogio, Chiara论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAKohler, Jens论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAZhou, Zhi-Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAWang, Haiyun论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Sch Life Sci & Technol, Shanghai 200092, Peoples R China Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA论文数: 引用数: h-index:机构:Li, Jiaqi论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Li, Shuai论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USALv, Qi论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Sch Life Sci & Technol, Shanghai 200092, Peoples R China Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAGondi, Sudershan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAHunter, John C.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USALu, Jia论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA论文数: 引用数: h-index:机构:Santamaria, David论文数: 0 引用数: 0 h-index: 0机构: Univ Bordeaux, INSERM, U1218, ACT Lab,IECB, F-33600 Pessac, France Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAWestover, Kenneth D.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Belfer Ctr Appl Canc Sci, Boston, MA 02215 USA Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA
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- [45] KRAS inhibitor found after decades of searchingFUTURE MEDICINAL CHEMISTRY, 2013, 5 (16) : 1907 - 1907Parks, Lisa论文数: 0 引用数: 0 h-index: 0
- [46] An allosteric pan-TEAD inhibitor blocks oncogenic YAP/TAZ signaling and overcomes KRAS G12C inhibitor resistanceNature Cancer, 2023, 4 : 812 - 828Thijs J. Hagenbeek论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyJason R. Zbieg论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMarc Hafner论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyRana Mroue论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyJennifer A. Lacap论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyNicole M. Sodir论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyCameron L. Noland论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyShervin Afghani论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyAyush Kishore论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyKamakoti P. Bhat论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyXiaosai Yao论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyStephen Schmidt论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologySaundra Clausen论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMicah Steffek论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyWendy Lee论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyPaul Beroza论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyScott Martin论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyEva Lin论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyRina Fong论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyPaola Di Lello论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMarta H. Kubala论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMichelle N.-Y. Yang论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyJeffrey T. Lau论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyEmily Chan论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyAlfonso Arrazate论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyLe An论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyElizabeth Levy论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMaria N. Lorenzo论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyHo-June Lee论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyTrang H. Pham论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyZora Modrusan论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyRichard Zang论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyYi-Chen Chen论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMichal Kabza论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMusaddeque Ahmed论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyJason Li论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMatthew T. Chang论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyDanilo Maddalo论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyMarie Evangelista论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyXin Ye论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyJames J. Crawford论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery OncologyAnwesha Dey论文数: 0 引用数: 0 h-index: 0机构: Genentech,Department of Discovery Oncology
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A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USASodir, Nicole M. M.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USANoland, Cameron L. L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Struct Biol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAAfghani, Shervin论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAKishore, Ayush论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USABhat, Kamakoti P. P.论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAYao, Xiaosai论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Oncol Bioinformat, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USASchmidt, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAClausen, Saundra论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USASteffek, Micah论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USALee, Wendy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USABeroza, Paul论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAMartin, Scott论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USALin, Eva论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAFong, Rina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Struct Biol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USADi Lello, Paola论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Struct Biol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAKubala, Marta H. H.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Struct Biol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAYang, Michelle N. -Y.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USALau, Jeffrey T. 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N.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Prot Chem, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USALee, Ho-June论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAPham, Trang H. H.论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAModrusan, Zora论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Microchem Prote & Lipid, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAZang, Richard论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAChen, Yi-Chen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAKabza, Michal论文数: 0 引用数: 0 h-index: 0机构: Roche Polska, Warsaw, Poland Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAAhmed, Musaddeque论文数: 0 引用数: 0 h-index: 0机构: Roche Canada, Mississauga, ON, Canada Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USALi, Jason论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Oncol Bioinformat, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAChang, Matthew T. T.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Oncol Bioinformat, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAMaddalo, Danilo论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAEvangelista, Marie论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USAYe, Xin论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USACrawford, James J. J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USADey, Anwesha论文数: 0 引用数: 0 h-index: 0机构: Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA Dept Discovery Oncol, Genentech, San Francisco, CA 94080 USA
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