首页
学术期刊
论文检测
AIGC检测
热点
更多
数据
Cyclin E1 protein overexpression sensitizes ovarian cancer cells to ZN-c3, a novel, selective and oral bioavailable inhibitor of Wee1
被引:4
|
作者
:
Ma, Jianhui
论文数:
0
引用数:
0
h-index:
0
Ma, Jianhui
Liu, Wen
论文数:
0
引用数:
0
h-index:
0
Liu, Wen
Chung, Heekyung
论文数:
0
引用数:
0
h-index:
0
Chung, Heekyung
Izadi, Hooman
论文数:
0
引用数:
0
h-index:
0
Izadi, Hooman
DeJong, Petrus
论文数:
0
引用数:
0
h-index:
0
DeJong, Petrus
Harismendy, Olivier
论文数:
0
引用数:
0
h-index:
0
Harismendy, Olivier
Li, Jia
论文数:
0
引用数:
0
h-index:
0
Li, Jia
Donate, Fernando
论文数:
0
引用数:
0
h-index:
0
Donate, Fernando
Samatar, Ahmed
论文数:
0
引用数:
0
h-index:
0
Samatar, Ahmed
Lackner, Mark
论文数:
0
引用数:
0
h-index:
0
Lackner, Mark
Escoubet, Laure
论文数:
0
引用数:
0
h-index:
0
Escoubet, Laure
Bunker, Kevin
论文数:
0
引用数:
0
h-index:
0
Bunker, Kevin
Kim, Daehwan
论文数:
0
引用数:
0
h-index:
0
Kim, Daehwan
Jameson, Nathan
论文数:
0
引用数:
0
h-index:
0
Jameson, Nathan
Ozmen, Tugba Yildiran
论文数:
0
引用数:
0
h-index:
0
Ozmen, Tugba Yildiran
Jeong, Kangjin
论文数:
0
引用数:
0
h-index:
0
Jeong, Kangjin
Zhang, Dong
论文数:
0
引用数:
0
h-index:
0
Zhang, Dong
Pan, Wen-An
论文数:
0
引用数:
0
h-index:
0
Pan, Wen-An
Mills, Gordon
论文数:
0
引用数:
0
h-index:
0
Mills, Gordon
机构
:
来源
:
CANCER RESEARCH
|
2023年
/ 83卷
/ 07期
关键词
:
D O I
:
10.1158/1538-7445.AM2023-2153
中图分类号
:
R73 [肿瘤学];
学科分类号
:
100214 ;
摘要
:
2153
引用
收藏
页数:3
相关论文
共 50 条
[11]
Clinical activity of single-agent ZN-c3, an oral WEE1 inhibitor, in a phase 1 dose-escalation trial in patients with advanced solid tumors.
Tolcher, Anthony
论文数:
0
引用数:
0
h-index:
0
机构:
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Tolcher, Anthony
Mamdani, Hirva
论文数:
0
引用数:
0
h-index:
0
机构:
Karmanos Canc Ctr, Detroit, MI USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Mamdani, Hirva
Chalasani, Pavani
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Arizona, Ctr Canc, Tucson, AZ USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Chalasani, Pavani
Meric-Bernstam, Funda
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Meric-Bernstam, Funda
Gazdoiu, Mihaela
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Gazdoiu, Mihaela
Makris, Lukas
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Makris, Lukas
Pultar, Philippe
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Pultar, Philippe
Voliotis, Dimitris
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Texas Oncol San Antonio Babcock, San Antonio, TX USA
Voliotis, Dimitris
CANCER RESEARCH,
2021,
81
(13)
[12]
BH3 mimetics synergize with the Wee1 inhibitor ZN-c3 by activating caspases which induce DNA damage and degrade key proteins
Izadi, Hooman
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Izadi, Hooman
Ibrahim, Noah
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Ibrahim, Noah
Hoang, Tiffany
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Hoang, Tiffany
Ma, Jianhui
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Ma, Jianhui
de Jong, Petrus R.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
de Jong, Petrus R.
Pinchman, Joseph
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Pinchman, Joseph
Bunker, Kevin D.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Bunker, Kevin D.
Samatar, Ahmed A.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Samatar, Ahmed A.
Donate, Fernando
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Donate, Fernando
CANCER RESEARCH,
2022,
82
(12)
[13]
Discovery of ZN-c3, a potent Wee-1 inhibitor with a differentiated pharmacologic and kinase selectivity profile.
Li, Jiali
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Li, Jiali
Boren, Brant
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Boren, Brant
Huang, Peter Q.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Huang, Peter Q.
Bunker, Kevin D.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Bunker, Kevin D.
Donate, Fernando
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Donate, Fernando
Samatar, Ahmed A.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Zentalis Pharmaceut, San Diego, CA USA
Samatar, Ahmed A.
CANCER RESEARCH,
2021,
81
(13)
[14]
A phase 1/2 dose escalation study of the BCL-2 inhibitor ZN-d5 and the WEE1 inhibitor azenosertib (ZN-c3) in patients (Pts) with acute myeloid leukemia (AML)
Smith, Catherine Choy
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Smith, Catherine Choy
Vachhani, Pankit
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Vachhani, Pankit
Garcia-Manero, Guillermo
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Garcia-Manero, Guillermo
Grieselhuber, Nicole Renee
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Grieselhuber, Nicole Renee
Murthy, Guru Subramanian Guru
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Murthy, Guru Subramanian Guru
Bhatia, Astha
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Bhatia, Astha
Arora, Jatinder
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Arora, Jatinder
Izadi, Hooman
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Izadi, Hooman
Fiorino, Anthony
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Fiorino, Anthony
Rampal, Raajit
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Med, Div Hematol Oncol, San Francisco, CA 94143 USA
Rampal, Raajit
JOURNAL OF CLINICAL ONCOLOGY,
2023,
41
(16)
[15]
A novel, potent and selective inhibitor of Wee1 with robust antitumor activity in various cancer xenograph models
Gavory, Gerald
论文数:
0
引用数:
0
h-index:
0
Gavory, Gerald
O'Dowd, Colin
论文数:
0
引用数:
0
h-index:
0
O'Dowd, Colin
Burkamp, Frank
论文数:
0
引用数:
0
h-index:
0
Burkamp, Frank
Rountree, Shane
论文数:
0
引用数:
0
h-index:
0
Rountree, Shane
Rozycka, Ewelina
论文数:
0
引用数:
0
h-index:
0
Rozycka, Ewelina
Boyd, Caroline
论文数:
0
引用数:
0
h-index:
0
Boyd, Caroline
Gorges, Beronia
论文数:
0
引用数:
0
h-index:
0
Gorges, Beronia
Burton, Stephanie
论文数:
0
引用数:
0
h-index:
0
Burton, Stephanie
Wilkinson, Andy
论文数:
0
引用数:
0
h-index:
0
Wilkinson, Andy
Shepherd, Steven
论文数:
0
引用数:
0
h-index:
0
Shepherd, Steven
Janssen, Dominic
论文数:
0
引用数:
0
h-index:
0
Janssen, Dominic
McFarland, Mary
论文数:
0
引用数:
0
h-index:
0
McFarland, Mary
Rountree, Shane
论文数:
0
引用数:
0
h-index:
0
Rountree, Shane
Harrison, Tim
论文数:
0
引用数:
0
h-index:
0
Harrison, Tim
CANCER RESEARCH,
2016,
76
[16]
The WEE1 inhibitor AZD-1775 has synergic activity with trabectedin or lurbinectedin in ovarian cancer cells
Uboldi, Sarah
论文数:
0
引用数:
0
h-index:
0
Uboldi, Sarah
Carrassa, Laura
论文数:
0
引用数:
0
h-index:
0
Carrassa, Laura
Frapolli, Roberta
论文数:
0
引用数:
0
h-index:
0
Frapolli, Roberta
Ubezio, Paolo
论文数:
0
引用数:
0
h-index:
0
Ubezio, Paolo
Erba, Eugenio
论文数:
0
引用数:
0
h-index:
0
Erba, Eugenio
D'Incalci, Maurizio
论文数:
0
引用数:
0
h-index:
0
D'Incalci, Maurizio
CANCER RESEARCH,
2016,
76
[17]
Suppression of Sirt1 sensitizes lung cancer cells to WEE1 inhibitor MK-1775-induced DNA damage and apoptosis
G Chen
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
G Chen
B Zhang
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
B Zhang
H Xu
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
H Xu
Y Sun
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
Y Sun
Y Shi
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
Y Shi
Y Luo
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
Y Luo
H Jia
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
H Jia
F Wang
论文数:
0
引用数:
0
h-index:
0
机构:
Emory University School of Medicine,Department of Radiation Oncology
F Wang
Oncogene,
2017,
36
: 6863
-
6872
[18]
Combination of the BCL-2 inhibitor ZN-d5 with the WEE1 inhibitor ZN-c3 shows additive or synergistic anti-tumor activity in acute myeloid leukemia (AML) models
Izadi, Hooman
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Izadi, Hooman
Hoang, Tiffany
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Hoang, Tiffany
Ibrahim, Noah
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Ibrahim, Noah
Pinchman, Joseph
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Pinchman, Joseph
Boren, Brant C.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Boren, Brant C.
Ma, Jianhui
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Ma, Jianhui
de Jong, Petrus R.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
de Jong, Petrus R.
Li, Jiali
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Li, Jiali
Bunker, Kevin D.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Bunker, Kevin D.
Samatar, Ahmed A.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Samatar, Ahmed A.
Donate, Fernando
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis, San Diego, CA USA
Zentalis, San Diego, CA USA
Donate, Fernando
CANCER RESEARCH,
2022,
82
(12)
[19]
Suppression of Sirt1 sensitizes lung cancer cells to WEE1 inhibitor MK-1775-induced DNA damage and apoptosis
Chen, G.
论文数:
0
引用数:
0
h-index:
0
机构:
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Chen, G.
Zhang, B.
论文数:
0
引用数:
0
h-index:
0
机构:
Xi An Jiao Tong Univ, Dept Physiol & Pathophysiol, Sch Med, Xian, Shaanxi, Peoples R China
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Zhang, B.
Xu, H.
论文数:
0
引用数:
0
h-index:
0
机构:
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Xu, H.
Sun, Y.
论文数:
0
引用数:
0
h-index:
0
机构:
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Sun, Y.
Shi, Y.
论文数:
0
引用数:
0
h-index:
0
机构:
Xidian Univ, Sch Life Sci & Technol, Engn Res Ctr Mol & Neuro Imaging, Minist Educ, Xian, Shaanxi, Peoples R China
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Shi, Y.
Luo, Y.
论文数:
0
引用数:
0
h-index:
0
机构:
Second Mil Med Univ, Changhai Hosp, Dept Neurosurg, Shanghai, Peoples R China
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Luo, Y.
Jia, H.
论文数:
0
引用数:
0
h-index:
0
机构:
Agr Univ Hebei, Dept Bioengn, Coll Food Sci & Technol, Baoding, Peoples R China
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Jia, H.
Wang, F.
论文数:
0
引用数:
0
h-index:
0
机构:
Xidian Univ, Sch Life Sci & Technol, Engn Res Ctr Mol & Neuro Imaging, Minist Educ, Xian, Shaanxi, Peoples R China
Emory Univ, Sch Med, Dept Radiat Oncol, Atlanta, GA 30322 USA
Wang, F.
ONCOGENE,
2017,
36
(50)
: 6863
-
6872
[20]
ZN-c3, a potent and selective Wee-1 inhibitor demonstrates anti-tumor activities in combination with other targeted therapies and overcomes PARP inhibitor resistance
Li, Jiali
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Li, Jiali
Ma, Jianhui
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Ma, Jianhui
de Jong, Petrus R.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
de Jong, Petrus R.
Izadi, Hooman
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Izadi, Hooman
Hoang, Tiffany
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Hoang, Tiffany
Ibrahim, Noah
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Ibrahim, Noah
Boren, Brant
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Boren, Brant
Hegde, Sayee Hegde
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Hegde, Sayee Hegde
Donate, Fernando
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, San Diego, CA USA
Zentalis Pharmaceut, San Diego, CA USA
Donate, Fernando
Samatar, Ahmed A.
论文数:
0
引用数:
0
h-index:
0
机构:
Zentalis Pharmaceut, New York, NY USA
Zentalis Pharmaceut, San Diego, CA USA
Samatar, Ahmed A.
CANCER RESEARCH,
2022,
82
(12)
←
1
2
3
4
5
→